SCHEMBL7477441

SCHEMBL7477441

CC(C)(C)OC(=O)C1(CN2C(=O)c3cccnc3C2=O)Cc2cc(N)sc2CO1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
TSHR P16473 1/20 0.36
KDM4E B2RXH2 1/20 0.36
TP53 P04637 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CA1 P00915 3/20 0.35
CA2 P00918 3/20 0.35
HPGD P15428 1/20 0.35
KMT2A Q03164 2/20 0.34
RXFP1 Q9HBX9 3/20 0.33
HDAC1 Q13547 1/20 0.33
HCRTR1 O43613 1/20 0.33
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7473201 0.81 AKT1 (0.30)
SCHEMBL7476167 0.76 ALDH1A1 (0.30) ALDH1A1GAA
SCHEMBL7468914 0.76 ALDH1A1 (0.30) ALDH1A1GAA
SCHEMBL7479494 0.76
SCHEMBL7466109 0.72
SCHEMBL7464864 0.70 KDM4E (0.34) KDM4ESMN1; SMN2
SCHEMBL5838384 0.66 ALDH1A1 (0.35) ALDH1A1L3MBTL1TSHRKDM4ETP53
SCHEMBL7474476 0.63 PDE4D (0.32)
SCHEMBL7471265 0.62 ACHE (0.31) L3MBTL1SMN1; SMN2HPGDKMT2AMEN1
SCHEMBL11872791 0.61 CYP1A2 (0.59) ALDH1A1L3MBTL1TSHRKDM4ETP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214325-A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases) NOVO NORDISK A/S (DK) 2002-06-19 EP disclosed
WO-2001019831-A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases) NOVO NORDISK A/S (DK) 2001-03-22 WO disclosed