SCHEMBL7480910

SCHEMBL7480910

NC(=O)Oc1cccc2[nH]c(-c3c(CCCCN4C(=O)c5ccccc5C4=O)[nH]c4ccccc34)nc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
MAPT P10636 3/20 0.41
NPSR1 Q6W5P4 2/20 0.41
HSD17B10 Q99714 2/20 0.40
HPGD P15428 1/20 0.40
MAPK1 P28482 1/20 0.40
PARP1 P09874 2/20 0.38
PKM P14618 1/20 0.37
TDP1 Q9NUW8 2/20 0.37
GPR84 Q9NQS5 1/20 0.36
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
DHODH Q02127 1/20 0.35
CYP1B1 Q16678 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
HDAC8 Q9BY41 3/20 0.34
HDAC3 O15379 2/20 0.34
HDAC4 P56524 2/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC7 Q8WUI4 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6584637 0.76 PARP1 (0.39) ALDH1A1MAPTNPSR1PARP1DHODH
SCHEMBL6587182 0.74 MEN1 (0.52) ALDH1A1MAPTNPSR1HSD17B10HPGD
SCHEMBL6585095 0.71 DHODH (0.47) PARP1DHODH
SCHEMBL6586959 0.69 KDM4E (0.56) ALDH1A1MAPTHSD17B10HPGDPARP1
SCHEMBL6588173 0.69 PARP1 (0.49) ALDH1A1PARP1KMT2AMEN1DHODH
Acetic Acid SCHEMBL7823040 0.67 ALDH1A1 (0.45) ALDH1A1MAPTNPSR1HSD17B10HPGD
SCHEMBL6587303 0.67 EPHX2 (0.52) PARP1DHODH
SCHEMBL6587773 0.66 PARP1 (0.46) ALDH1A1MAPTHSD17B10HPGDPARP1
SCHEMBL6588299 0.65 PARP1 (0.47) ALDH1A1MAPTNPSR1PARP1L3MBTL1
SCHEMBL6578295 0.64 PARP1 (0.52) ALDH1A1PARP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-02-06 EP disclosed
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed
WO-2000068206-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2000-11-16 WO disclosed