SCHEMBL6584637

SCHEMBL6584637

CCCC(c1[nH]c2ccccc2c1-c1nc2c(OC(N)=O)cccc2[nH]1)N1C(=O)c2ccccc2C1=O

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.39
DHODH Q02127 1/20 0.36
ALDH1A1 P00352 4/20 0.35
KDM4E B2RXH2 2/20 0.35
GAA P10253 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
RXFP1 Q9HBX9 1/20 0.35
TNF P01375 4/20 0.35
ADORA1 P30542 1/20 0.34
GSK3B P49841 1/20 0.34
ADK P55263 1/20 0.34
PDE4A P27815 3/20 0.33
PDE4B Q07343 3/20 0.33
PDE4C Q08493 3/20 0.33
PDE4D Q08499 3/20 0.33
MAPT P10636 2/20 0.33
CBFB Q13951 1/20 0.33
PDE5A O76074 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6805765 0.87 PARP1 (0.50) PARP1DHODH
SCHEMBL6805769 0.79 KDM4E (0.37) PARP1ALDH1A1KDM4EGAANPSR1
SCHEMBL7480910 0.76 ALDH1A1 (0.41) PARP1DHODHALDH1A1NPSR1MAPT
SCHEMBL6587182 0.75 MEN1 (0.52) PARP1DHODHALDH1A1KDM4ENPSR1
SCHEMBL6586959 0.70 KDM4E (0.56) PARP1ALDH1A1KDM4EMAPT
SCHEMBL6585095 0.70 DHODH (0.47) PARP1DHODHGAA
SCHEMBL6587303 0.68 EPHX2 (0.52) PARP1DHODH
SCHEMBL6588173 0.68 PARP1 (0.49) PARP1DHODHALDH1A1PDE5A
SCHEMBL6578295 0.67 PARP1 (0.52) PARP1ALDH1A1KDM4EPDE4APDE4B
SCHEMBL6589817 0.67 PIM1 (0.41) PARP1ALDH1A1KDM4EGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed