SCHEMBL7483897

SCHEMBL7483897

O=C(O)c1ccccc1Cc1cc2cc(-c3ccc(F)cc3)ccc2[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 1/20 0.45
DHODH Q02127 4/20 0.41
PCSK9 Q8NBP7 2/20 0.41
TSHR P16473 2/20 0.41
KDM4E B2RXH2 1/20 0.41
PDPK1 O15530 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 1/20 0.41
NFKB1 P19838 1/20 0.41
APEX1 P27695 1/20 0.41
CYP2C19 P33261 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
DCLRE1B Q9H816 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
DCLRE1A Q6PJP8 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7477639 0.89 TSHR (0.51) F2DHODHTSHRKDM4EALDH1A1
SCHEMBL7475485 0.79 MMP12 (0.42) F2TSHRKDM4EALDH1A1NFKB1
SCHEMBL7482853 0.77 HRH3 (0.50) F2TSHRKDM4EALDH1A1LMNA
SCHEMBL7478027 0.73 ALDH1A1 (0.48) TSHRKDM4EALDH1A1LMNAHSD17B10
SCHEMBL20494483 0.72 KDM4E (0.76) TSHRKDM4EPDPK1ALDH1A1LMNA
SCHEMBL7474003 0.71 HRH3 (0.60) F2TSHRKDM4EALDH1A1LMNA
SCHEMBL12597050 0.71 PPARG (0.55) TSHRLMNANPC1GPR17
SCHEMBL7474368 0.71 KDM4E (0.52) KDM4EALDH1A1HPGDHSD17B10
SCHEMBL19953414 0.70 LOXL2 (0.57) PCSK9
SCHEMBL4872353 0.70 TSHR (0.72) TSHRALDH1A1HPGDCYP2C19CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1210343-A2 BENZOIC ACID DERIVATIVES AND THEIR USE AS PPAR RECEPTOR AGONISTS AstraZeneca AB (SE) 2002-06-05 EP disclosed
WO-2001012187-A2 BENZOIC ACID DERIVATIVES AND THEIR USE AS PPAR RECEPTOR AGONISTS ASTRAZENECA AB (SE) 2001-02-22 WO disclosed