SCHEMBL749300

SCHEMBL749300

CC(C)(C)c1ccc(CN(CCc2ccc3c(c2)OCO3)C(=O)c2cccc3c2NCCC3)cc1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
MAPT P10636 2/20 0.40
HPGD P15428 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
TSHR P16473 3/20 0.36
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
PKM P14618 1/20 0.36
ALOX15 P16050 1/20 0.36
ALOX12 P18054 1/20 0.36
HSD17B10 Q99714 1/20 0.36
LMNA P02545 1/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL748464 0.89 ALDH1A1 (0.37) ALDH1A1MAPTHPGDSMN1; SMN2NPSR1
SCHEMBL749367 0.86 ALDH1A1 (0.40) ALDH1A1MAPTSMN1; SMN2NPSR1TSHR
SCHEMBL745473 0.86 KMT2A (0.44) MAPT
SCHEMBL748523 0.86 LPAR1 (0.38)
SCHEMBL748780 0.86 TP53 (0.35) ALDH1A1MAPTKDM4E
SCHEMBL745501 0.86 TMEM97 (0.39) ALDH1A1TSHR
SCHEMBL748724 0.86 F10 (0.40)
SCHEMBL748461 0.85 ESRRG (0.46) MAPTPKMLMNA
Hydrochloric Acid SCHEMBL752637 0.85 TMEM97 (0.38) ALDH1A1TSHR
SCHEMBL747130 0.85 SLC13A5 (0.37) MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049493-B1 COMPOUNDS SUITABLE AS MODULATORS OF HDL CADILA HEALTHCARE LTD (IN) 2012-03-21 EP disclosed
US-8022217-B2 Compounds suitable as modulators of HDL CADILA HEALTHCARE LIMITED (IN) 2011-09-20 US disclosed