SCHEMBL7514977

SCHEMBL7514977

O=C(N[C@H]1CCOC1O)[C@H](Cc1ccccc1)NC(=S)Cc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 14/20 0.59
ALDH1A1 P00352 1/20 0.43
CAPNS1 P04632 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8810989 0.89 CAPN1 (0.75) CAPN1CAPNS1
SCHEMBL8812573 0.82 CTSK (0.60) CAPN1
SCHEMBL8812581 0.82 CTSK (0.60) CAPN1
SCHEMBL27427437 0.80 CTSS (0.56) CAPN1
SCHEMBL7516532 0.80 CTSS (0.56) CAPN1
SCHEMBL7514986 0.80 CAPN1 (0.52) CAPN1ALDH1A1CAPNS1
SCHEMBL7517586 0.80 CAPN1 (0.54) CAPN1CAPNS1
SCHEMBL7514607 0.77 CAPN1 (0.49) CAPN1ALDH1A1
SCHEMBL7514760 0.75 CAPN1 (0.49) CAPN1CAPNS1
SCHEMBL4972757 0.74 CAPN1 (1.00) CAPN1CAPNS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP claimed
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP disclosed