SCHEMBL7517586

SCHEMBL7517586

O=C(N[C@H]1CCOC1O)C(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 17/20 0.54
CYP1A2 P05177 1/20 0.42
CAPNS1 P04632 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7514977 0.80 CAPN1 (0.59) CAPN1CAPNS1
SCHEMBL8812573 0.79 CTSK (0.60) CAPN1
SCHEMBL8812581 0.79 CTSK (0.60) CAPN1
SCHEMBL7516532 0.78 CTSS (0.56) CAPN1
SCHEMBL17852711 0.76 ALDH1A1 (0.54) CAPN1
SCHEMBL21006007 0.75 CAPN1 (0.48) CAPN1CYP1A2CAPNS1
SCHEMBL21880812 0.75 EPHX2 (0.58) CAPN1
SCHEMBL7514607 0.74 CAPN1 (0.49) CAPN1
SCHEMBL8810080 0.74 CAPN1 (0.62) CAPN1CYP1A2
SCHEMBL8810071 0.74 CAPN1 (0.62) CAPN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP claimed
US-5496834-A PEPTIDE DERIVATIVES AS CATHEPSIN L INHIBITORS AND INHIBITORS OF BONE RESORPTION OR TREATMENT OF OSTEOPOROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-03-05 US claimed
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP disclosed