SCHEMBL7527286

SCHEMBL7527286

COc1ccc(C(=O)n2ccc(NCC(=O)O)nc2=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.43
KMT2A Q03164 4/20 0.41
ALDH1A1 P00352 1/20 0.41
KLK7 P49862 1/20 0.41
KLK14 Q9P0G3 1/20 0.41
KLK5 Q9Y337 1/20 0.41
ELANE P08246 1/20 0.39
PTGER2 P43116 2/20 0.39
PTGS1 P23219 1/20 0.38
HPGD P15428 1/20 0.38
POLB P06746 1/20 0.38
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
UBE2N P61088 1/20 0.38
KDM4E B2RXH2 1/20 0.38
TSHR P16473 1/20 0.38
PDE4B Q07343 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5983023 0.76 KMT2A (0.55) KMT2AALDH1A1KLK7KLK14KLK5
SCHEMBL9335990 0.70 CTRB1 (0.39) KMT2AALDH1A1
SCHEMBL7528362 0.69 ADORA3 (0.51) KMT2AALDH1A1KDM4E
SCHEMBL6886945 0.67 KMT2A (0.50) KMT2AALDH1A1KLK7KLK14KLK5
Hydrochloric Acid SCHEMBL3655605 0.67 MAPT (0.59) PTGS2KMT2AALDH1A1POLBCA1
SCHEMBL1797197 0.67 MAPT (0.59) PTGS2KMT2AALDH1A1POLBCA1
SCHEMBL6880479 0.66 KMT2A (0.52) KMT2AALDH1A1KLK7KLK14KLK5
SCHEMBL12882191 0.65 KMT2A (0.51) KMT2AALDH1A1KLK7KLK14KLK5
SCHEMBL2796671 0.64 ALDH1A1 (0.67) KMT2AALDH1A1HPGDPOLBCA1
Hydrochloric Acid SCHEMBL3246059 0.63 LMNA (0.65) KMT2AALDH1A1POLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0761681-B1 Process for the preparation of substituted derivatives of N-ethylglycine HOECHST AG (DE) 2002-03-13 EP disclosed