SCHEMBL7537367

SCHEMBL7537367

COc1ccc(-c2nnc(C(=O)CCCCNC(=O)C3(C(N)=O)CCCCC3)o2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.42
CTSL P07711 1/20 0.42
CTSB P07858 1/20 0.42
CTSS P25774 1/20 0.42
HDAC8 Q9BY41 2/20 0.42
CES1 P23141 2/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
CACNA1B Q00975 1/20 0.40
APBA1 Q02410 1/20 0.40
HSD17B10 Q99714 1/20 0.40
HDAC1 Q13547 4/20 0.40
HDAC6 Q9UBN7 4/20 0.40
HTT P42858 1/20 0.39
FAAH O00519 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7647908 0.78 CTSL (0.68) CTSKCTSLCTSBCTSS
SCHEMBL7528404 0.78 CTSL (0.35) CTSKCTSLCTSBCTSSCES1
SCHEMBL7560363 0.78 CTSS (0.64) CTSKCTSLCTSBCTSSHTT
SCHEMBL7537370 0.73 POLB (0.40) CTSKCTSLCTSBCTSSHDAC8
SCHEMBL7533228 0.72 DAGLA (0.50) CTSSHDAC8CES1HDAC1HDAC6
SCHEMBL7530434 0.72 DAGLA (0.52) HDAC8CES1HDAC1HDAC6FAAH
SCHEMBL7537340 0.70 CTSL (0.66) CTSKCTSLCTSBCTSSCES1
SCHEMBL7560369 0.69 CTSS (0.67) CTSKCTSLCTSBCTSSHTT
SCHEMBL30968135 0.68 NPC1 (0.61) HDAC8KMT2AKDM4EALDH1A1HPGD
SCHEMBL30968155 0.67 SMPD1 (0.61) HDAC8KMT2AKDM4EALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002023784-A2 CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2002-03-21 WO disclosed