SCHEMBL7544301

SCHEMBL7544301

COc1ccc(Br)c2c1C=CCC2

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.46
CYP1A2 P05177 1/20 0.39
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
CYP19A1 P11511 1/20 0.34
NQO2 P16083 2/20 0.33
ERN1 O75460 1/20 0.33
ALDH1A1 P00352 2/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
DRD2 P14416 4/20 0.32
DRD1 P21728 4/20 0.32
ADRA1A P35348 2/20 0.32
BCHE P06276 1/20 0.31
ACHE P22303 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HTR2B P41595 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8670294 0.85 KDM4E (0.40) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL2970791 0.82 KDM4E (0.45) KDM4ECYP1A2HDAC1HDAC6CYP19A1
SCHEMBL7543660 0.77 KDM4E (0.39) KDM4EALDH1A1GAAHPGD
SCHEMBL7540968 0.77 HTR2A (0.47) KDM4EHTR2AHTR2CHTR2B
SCHEMBL7548030 0.76 ALDH1A1 (0.32) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL7548035 0.76 ADORA3 (0.31) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL7551757 0.73 HTR2A (0.43) KDM4ECYP1A2ALDH1A1HTR2AHTR2C
SCHEMBL2974200 0.71 KDM4E (0.41) KDM4ECYP1A2HDAC1HDAC6CYP19A1
SCHEMBL15056458 0.71 KDM4E (0.45) KDM4ECYP1A2HDAC1HDAC6CYP19A1
SCHEMBL8908569 0.70 ADRA1A (0.42) KDM4EALDH1A1GLAGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0883599-B1 AMINOTETRALIN DERIVATIVES AND COMPOSITIONS AND METHOD OF USE THEREOF ASTRAZENECA AB (SE) 2002-06-05 EP disclosed
EP-0883599-A1 AMINOTETRALIN DERIVATIVES AND COMPOSITIONS AND METHOD OF USE THEREOF ZENECA LIMITED (GB) 1998-12-16 EP disclosed
US-5807897-A MUSCULAR DISORDERS ZENECA LIMITED (GB) 1998-09-15 US disclosed
WO-1997031887-A1 AMINOTETRALIN DERIVATIVES AND COMPOSITIONS AND METHOD OF USE THEREOF ZENECA LIMITED (GB) 1997-09-04 WO disclosed