SCHEMBL7546700

SCHEMBL7546700

Cc1occc1CC(=O)c1ccnc(N)c1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.39
NAPRT Q6XQN6 1/20 0.35
L3MBTL1 Q9Y468 4/20 0.33
KMT2A Q03164 3/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
CYP2C19 P33261 2/20 0.33
KDM4E B2RXH2 2/20 0.33
GAA P10253 1/20 0.33
PKM P14618 1/20 0.33
TDP1 Q9NUW8 2/20 0.32
TP53 P04637 2/20 0.32
ESR1 P03372 1/20 0.32
POLB P06746 1/20 0.32
APEX1 P27695 1/20 0.32
MAPK1 P28482 1/20 0.32
ESR2 Q92731 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7548395 0.89 ALOX5 (0.38) ALOX5L3MBTL1NPC1RAB9ASMN1; SMN2
SCHEMBL7546681 0.82 TDP1 (0.37) NAPRTL3MBTL1KMT2ASMN1; SMN2KDM4E
SCHEMBL7547894 0.81 MAPT (0.46) NAPRTKMT2AKDM4EMEN1
SCHEMBL7543322 0.79 KMT2A (0.41) NAPRTL3MBTL1KMT2ANPC1RAB9A
SCHEMBL9059311 0.79 NAPRT (0.34) NAPRTKMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL7551790 0.77 SGMS2 (0.36) NAPRTKDM4ETP53POLBMAPK1
SCHEMBL8805065 0.75 SHBG (0.44) NAPRTKMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL8799100 0.73 KDM4E (0.44) ALOX5NAPRTKMT2ANPC1RAB9A
SCHEMBL7551656 0.72 TDP1 (0.39) NAPRTL3MBTL1KMT2ANPC1RAB9A
SCHEMBL19857454 0.72 NAPRT (0.57) NAPRTL3MBTL1KMT2ARAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997049708-A9 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS 1998-05-22 WO disclosed