SCHEMBL755183

SCHEMBL755183

O=C(O)N1CCOc2ccc(Oc3cccc(-c4ncco4)c3)cc2S1(=O)=O

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 10/20 0.41
MGLL Q99685 1/20 0.38
GPR142 Q7Z601 2/20 0.37
FAAH O00519 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL782067 0.88 BACE1 (0.38) LTA4HMGLLGPR142FAAH
SCHEMBL757503 0.83 PIK3CD (0.36) GPR142FAAH
SCHEMBL760502 0.83 FFAR1 (0.38) GPR142FAAH
SCHEMBL759900 0.82 FAAH (0.44) GPR142FAAH
SCHEMBL756393 0.79 GPR142 (0.38) MGLLGPR142FAAH
SCHEMBL755478 0.79 LMNA (0.46) GPR142
SCHEMBL757739 0.78 KEAP1 (0.43) LTA4HMGLLFAAH
SCHEMBL759673 0.75 MAPT (0.43) FAAH
SCHEMBL782015 0.72 GPR119 (0.38)
SCHEMBL758615 0.72 TDP1 (0.45) FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2431360-B1 Derivatives of dihydrobenzoxathiazepine, method of preparing same and pharmaceutical compositions containing them as well as their uses as modulators of AMPA receptors SERVIER LAB (FR) 2013-04-17 EP disclosed
EP-2431360-A1 Derivatives of dihydrobenzoxathiazepine, method of preparing same and pharmaceutical compositions containing them as well as their uses as modulators of AMPA receptors Les Laboratoires Servier (FR) 2012-03-21 EP disclosed