SCHEMBL7554022

SCHEMBL7554022

COc1ccc(-c2ccc(-c3nc4ccc(OC)cc4c(=O)n3CCCN)s2)c(OC)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F11 P03951 1/20 0.50
RXRA P19793 1/20 0.44
TDP1 Q9NUW8 6/20 0.42
CRHR1 P34998 3/20 0.41
P2RX3 P56373 1/20 0.41
HSP90AA1 P07900 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
DYRK1A Q13627 2/20 0.40
HASPIN Q8TF76 2/20 0.40
DYRK3 O43781 1/20 0.40
CLK1 P49759 1/20 0.40
CLK2 P49760 1/20 0.40
CLK3 P49761 1/20 0.40
GSK3B P49841 1/20 0.40
DYRK2 Q92630 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
DYRK4 Q9NR20 1/20 0.40
DYRK1B Q9Y463 1/20 0.40
MPO P05164 1/20 0.39
PDE4A P27815 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6313495 0.95 F11 (0.46) F11RXRATDP1CRHR1P2RX3
SCHEMBL6314138 0.94 F11 (0.45) F11RXRATDP1CRHR1
SCHEMBL6313995 0.93 RXRA (0.52) RXRATDP1HSP90AA1NPSR1KDM4E
SCHEMBL6307883 0.88 EGFR (0.46) F11RXRATDP1CRHR1CYP3A4
SCHEMBL6306810 0.85 F11 (0.62) F11RXRATDP1KDM4E
SCHEMBL6308042 0.84 F11 (0.49) F11RXRANPSR1DYRK1AHASPIN
SCHEMBL6313461 0.83 F11 (0.41) F11TDP1HSP90AA1NPSR1CYP1A2
SCHEMBL7549056 0.83 F11 (0.59) F11RXRATDP1P2RX3KDM4E
SCHEMBL6308861 0.81 F11 (0.57) F11RXRATDP1P2RX3KDM4E
SCHEMBL5877056 0.81 CRHR1 (0.43) F11CRHR1P2RX3HSP90AA1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216235-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023365-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed