SCHEMBL755449

SCHEMBL755449

CC1(C)Oc2cc([N+](=O)[O-])ccc2N(c2ccccc2F)C1c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.45
HTT P42858 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.39
MAPT P10636 6/20 0.39
TNKS O95271 3/20 0.37
KMT2A Q03164 4/20 0.36
MEN1 O00255 3/20 0.36
GAA P10253 2/20 0.36
MAPK1 P28482 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
CCKBR P32239 1/20 0.36
GABRA3 P34903 1/20 0.36
OPRK1 P41145 1/20 0.36
MC3R P41968 1/20 0.36
GABRA2 P47869 1/20 0.36
GABRB2 P47870 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2265909 0.87 HTT (0.42) ALDH1A1HTTL3MBTL1MAPTTNKS
SCHEMBL27735508 0.72 L3MBTL1 (0.41) ALDH1A1HTTL3MBTL1MAPTKMT2A
SCHEMBL755966 0.68 TNKS (0.45) TNKSHSD11B1
SCHEMBL27756121 0.67 ALDH1A1 (0.35) ALDH1A1HTTL3MBTL1MAPTKMT2A
SCHEMBL758334 0.66 ALDH1A1 (0.41) ALDH1A1HTTL3MBTL1MAPTKMT2A
SCHEMBL27735521 0.66 WDR5 (0.39) ALDH1A1HTTMAPTKMT2AMEN1
SCHEMBL27735510 0.65 CASP1 (0.43) ALDH1A1L3MBTL1MAPTKMT2AMEN1
SCHEMBL754188 0.65 MAPT (0.46) ALDH1A1HTTL3MBTL1MAPTKMT2A
SCHEMBL27735485 0.65 NFE2L2 (0.40) ALDH1A1HTTL3MBTL1MAPTKMT2A
SCHEMBL3039656 0.61 CASP1 (0.47) ALDH1A1HTTL3MBTL1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1984345-B9 BENZOXAZINES AND RELATED NITROGEN-CONTAINING HETEROBICYCLIC COMPOUNDS USEFUL AS MINERALOCORTICOID RECEPTOR MODULATING AGENTS MITSUBISHI TANABE PHARMA CORP (JP) 2012-03-21 EP disclosed
EP-1984345-B1 BENZOXAZINES AND RELATED NITROGEN-CONTAINING HETEROBICYCLIC COMPOUNDS USEFUL AS MINERALOCORTICOID RECEPTOR MODULATING AGENTS MITSUBISHI TANABE PHARMA CORP (JP) 2011-08-31 EP disclosed