SCHEMBL7555544

SCHEMBL7555544

CC(C)CCc1cc(-c2c[nH]cn2)ccc1C(=O)NC(=O)NCC#N

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PRKD1 Q15139 2/20 0.34
CTSL P07711 5/20 0.33
CTSK P43235 3/20 0.33
ROCK2 O75116 1/20 0.32
ROCK1 Q13464 1/20 0.32
CTSB P07858 3/20 0.31
HTT P42858 1/20 0.31
JAK2 O60674 1/20 0.31
MAP4K4 O95819 1/20 0.31
CTSS P25774 3/20 0.31
SGK1 O00141 1/20 0.31
CAMKK2 Q96RR4 1/20 0.31
MAP1LC3B Q9GZQ8 1/20 0.31
MAP1LC3A Q9H492 1/20 0.31
BRS3 P32247 1/20 0.31
EGLN1 Q9GZT9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6183364 0.70 CTSB (0.35) CTSLCTSKCTSBHTTJAK2
SCHEMBL4701045 0.68 CTSK (0.45) CTSLCTSKCTSBCTSS
SCHEMBL6183366 0.66 NPC1 (0.40) PRKD1CTSKROCK2ROCK1CTSB
SCHEMBL2694733 0.65 SGK1 (0.51) SGK1CAMKK2
SCHEMBL5528914 0.60 ALDH1A1 (0.48) CTSLHTT
SCHEMBL21857189 0.59 KDM4E (0.50) ROCK2ROCK1JAK2
SCHEMBL5529215 0.59 ALDH1A1 (0.49) CTSLHTT
SCHEMBL11038741 0.57 KDM4E (0.53)
SCHEMBL5522997 0.57 SLC6A5 (0.48) HTT
SCHEMBL10912854 0.56 KDM4E (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1161415-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-12-12 EP disclosed
WO-2000055126-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO disclosed