SCHEMBL7557262

SCHEMBL7557262

OCc1ccncc1S.OCc1ccncc1SC(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.35
SLC22A12 Q96S37 8/20 0.33
APOBEC3G Q9HC16 1/20 0.33
KCNA5 P22460 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
HIF1A Q16665 1/20 0.32
GPBAR1 Q8TDU6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6233930 0.92 KIF11 (0.40) KIF11SLC22A12APOBEC3GKCNA5CYP1A2
SCHEMBL2643304 0.76
SCHEMBL864206 0.73 APOBEC3G (0.55) KIF11APOBEC3G
SCHEMBL6238584 0.64 ALDH1A1 (0.44) KIF11APOBEC3GCYP1A2CYP3A4CYP2C9
SCHEMBL1769946 0.62 CYP11B2 (0.53) SLC22A12KCNA5CYP1A2CYP3A4CYP2C9
SCHEMBL3078934 0.61 SLC22A12 (0.43) SLC22A12
SCHEMBL7557430 0.60 KCNA5 (0.42) KIF11KCNA5CYP1A2CYP3A4CYP2C9
SCHEMBL17318488 0.60 SCN9A (0.40) KIF11
SCHEMBL29900474 0.59 AOC1 (0.43)
SCHEMBL6249306 0.59 AOC1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222194-A1 7-ACYLAMINO-3-HETEROARYLTHIO-3-CEPHEM CARBOXYLIC ACID ANTIBIOTICS AND PRODRUGS THEREOF Essential Therapeutics, Inc. (US) 2002-07-17 EP disclosed
WO-2001021623-A1 7-ACYLAMINO-3-HETEROARYLTHIO-3-CEPHEM CARBOXYLIC ACID ANTIBIOTICS AND PRODRUGS THEREOF ESSENTIAL THERAPEUTICS, INC. (US) 2001-03-29 WO disclosed