SCHEMBL7562811

SCHEMBL7562811

CC1(C)C=CCC(c2ccc(F)c(F)c2)=C1

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PGR P06401 3/20 0.36
PTGS2 P35354 4/20 0.33
CREBBP Q92793 1/20 0.32
NOTUM Q6P988 1/20 0.31
PTGS1 P23219 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27456106 0.82 CYP11B1 (0.43)
SCHEMBL7543866 0.81 LPL (0.33) PTGS2PTGS1
SCHEMBL7624027 0.77 SIGMAR1 (0.34) PTGS2PTGS1
SCHEMBL19445334 0.69 NOTUM (0.41) PGRPTGS2CREBBPNOTUMPTGS1
SCHEMBL7568643 0.66 PGR (0.35) PGR
SCHEMBL13741967 0.63 CYP17A1 (0.52) PGRPTGS2NOTUMPTGS1
SCHEMBL31158855 0.62 CHRM5 (0.37) PGRPTGS2CREBBPNOTUMPTGS1
SCHEMBL7691782 0.61 CYP2A6 (0.35) PGR
SCHEMBL31158742 0.60 PTGS2 (0.35) PGRPTGS2CREBBPNOTUMPTGS1
SCHEMBL6816479 0.60 PCSK9 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1175411-A1 CYCLOTHIOCARBAMATE DERIVATIVES AS PROGESTERONE RECEPTOR MODULATORS American Home Products Corporation (US) 2002-01-30 EP disclosed
WO-2000066570-A1 CYCLOTHIOCARBAMATE DERIVATIVES AS PROGESTERONE RECEPTOR MODULATORS AMERICAN HOME PRODUCTS CORPORATION (US) 2000-11-09 WO disclosed