SCHEMBL7564537

SCHEMBL7564537

CCCCC(NC(=O)c1ccccc1)C(=O)CNS(=O)(=O)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.54
CASP1 P29466 1/20 0.47
LMNA P02545 2/20 0.46
PRSS1 P07477 2/20 0.46
CTSG P08311 2/20 0.46
CTRB1 P17538 2/20 0.46
CMA1 P23946 2/20 0.46
ALDH1A1 P00352 3/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA9 Q16790 2/20 0.43
EPHX2 P34913 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
HSD17B10 Q99714 1/20 0.43
MMP1 P03956 1/20 0.43
GAA P10253 1/20 0.43
MMP12 P39900 1/20 0.43
USP2 O75604 1/20 0.43
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7690188 0.89 EGFR (0.48) CA2
SCHEMBL7428250 0.85 KCNA5 (0.44) CA2CASP1EPHX2MMP1GAA
SCHEMBL7684139 0.85 CA2 (0.48) CA2LMNAALDH1A1CA12CA1
SCHEMBL7682470 0.84 ALDH1A1 (0.51) CA2LMNAALDH1A1GAA
SCHEMBL7675029 0.83 L3MBTL1 (0.44) CA2CASP1LMNAALDH1A1NPSR1
SCHEMBL7686060 0.83 EGFR (0.46) CA2
SCHEMBL7678439 0.82 ADAMTS4 (0.48) CA2CASP1LMNAMMP1GAA
SCHEMBL7680584 0.82 AKR1C3 (0.48) LMNAALDH1A1GAA
SCHEMBL7686484 0.82 CA2 (0.44) CA2CASP1CA12CA1CA9
SCHEMBL7695233 0.81 CAPN1 (0.54) CA2CASP1EPHX2MMP1MMP12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1073632-A1 SUBSTITUTED BENZAMIDES, THEIR PRODUCTION AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-02-07 EP disclosed
WO-1999054293-A1 SUBSTITUTED BENZAMIDES, THEIR PRODUCTION AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1999-10-28 WO disclosed