SCHEMBL7686484

SCHEMBL7686484

CCCCC(NC(=O)c1ccc(SCc2ccc3ccccc3c2)cc1)C(=O)CNS(=O)(=O)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.44
CCKBR P32239 1/20 0.42
DHFR P00374 4/20 0.41
FPGS Q05932 2/20 0.41
KAT6A Q92794 1/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
CASP1 P29466 1/20 0.37
POLB P06746 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA9 Q16790 1/20 0.37
LTB4R Q15722 1/20 0.37
ITGB1 P05556 1/20 0.36
ITGA4 P13612 1/20 0.36
PLA2G2A P14555 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7682464 0.91 CA2 (0.42) CA2CCKBRDHFRFPGSCTSL
SCHEMBL7704769 0.88 CA2 (0.52) CA2KAT6ACTSLCTSBCTSS
SCHEMBL7661370 0.87 CCKBR (0.44) CA2CCKBRDHFRFPGSCTSL
SCHEMBL7678439 0.86 ADAMTS4 (0.48) CA2CCKBRDHFRFPGSKAT6A
SCHEMBL7666410 0.85 CCKBR (0.42) CA2CCKBRDHFRFPGSCTSL
SCHEMBL7684139 0.84 CA2 (0.48) CA2CCKBRKAT6ACA12CA1
SCHEMBL7682470 0.82 ALDH1A1 (0.51) CA2CCKBRKAT6A
SCHEMBL7564537 0.82 CA2 (0.54) CA2CASP1CA12CA1CA9
SCHEMBL7701294 0.80 CA2 (0.50) CA2CTSLCTSBCTSSCTSK
SCHEMBL7680584 0.77 AKR1C3 (0.48) CCKBRKAT6AOPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436925-B1 BETTER ABLE TO CROSS MEMBRANES; INHIBITORS OF CYSTEINE PROTEASES LIKE CALPAIN I AND II AND CATHEPSIN B AND L, CAN THUS BE USED TO CONTROL DISEASES ASSOCIATED WITH AN ELEVATED ACTIVITY OF CALPAIN ENZYMES OR CATHEPSIN ENZYMES ABBOTT LABORATORIES 2002-08-20 US disclosed