SCHEMBL7572428

SCHEMBL7572428

CCOC(=O)c1ccc(NS(=O)(=O)c2cccc(Cl)c2C)c(NS(=O)(=O)c2cccc(Cl)c2C)c1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
KDM4E B2RXH2 2/20 0.54
LMNA P02545 1/20 0.54
TP53 P04637 1/20 0.51
HIF1A Q16665 1/20 0.47
HSD11B1 P28845 3/20 0.47
IKBKB O14920 1/20 0.47
CYP1A2 P05177 1/20 0.47
RAB9A P51151 1/20 0.47
HTT P42858 1/20 0.46
TSHR P16473 1/20 0.46
SLC40A1 Q9NP59 1/20 0.46
PKM P14618 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HSD17B1 P14061 1/20 0.45
HSD17B2 P37059 1/20 0.45
POLB P06746 1/20 0.44
MAPT P10636 1/20 0.44
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7573034 0.90 ACLY (0.53) ALDH1A1KDM4ETP53HSD11B1TSHR
SCHEMBL7577661 0.85 ALDH1A1 (0.49) ALDH1A1KDM4ELMNATP53HIF1A
SCHEMBL3777581 0.81 PTGES2 (0.65) ALDH1A1KDM4ELMNAHIF1AIKBKB
SCHEMBL7569885 0.78 ALDH1A1 (0.59) ALDH1A1TP53TSHRSLC40A1POLB
SCHEMBL7570489 0.78 LMNA (0.52) ALDH1A1KDM4ELMNATSHRSMN1; SMN2
SCHEMBL7588152 0.76 SLC40A1 (0.59) ALDH1A1TP53HSD11B1TSHRSLC40A1
SCHEMBL7594250 0.76 SLC40A1 (0.66) ALDH1A1HSD11B1SLC40A1PKMPOLB
SCHEMBL7594652 0.75 SLC40A1 (0.53) HSD11B1SLC40A1PKM
SCHEMBL7570349 0.74 ALDH1A1 (0.60) ALDH1A1KDM4ELMNAHIF1AHTT
SCHEMBL7578595 0.74 NPSR1 (0.72) ALDH1A1KDM4ELMNATP53HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1239852-A2 BISSULFONAMIDE DERIVATIVES AS ENZYME INHIBITORS Arrow Therapeutics Limited (GB) 2002-09-18 EP disclosed
WO-2001028537-A2 BISSULFONAMIDE DERIVATIVES AS ENZYME INHIBITORS ARROW THERAPEUTICS LIMITED (GB) 2001-04-26 WO disclosed