SCHEMBL7591337

SCHEMBL7591337

CCCOC(=O)c1cc(C(F)(F)F)c(F)c(F)c1F

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
PDK2 Q15119 1/20 0.40
LMNA P02545 2/20 0.39
TSHR P16473 4/20 0.38
TDP1 Q9NUW8 2/20 0.38
ESR1 P03372 2/20 0.38
CHRM1 P11229 1/20 0.38
SLC6A2 P23975 1/20 0.38
KDR P35968 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KDM4E B2RXH2 3/20 0.38
HSD17B10 Q99714 1/20 0.38
TP53 P04637 1/20 0.37
CYP3A4 P08684 1/20 0.37
MAPK1 P28482 1/20 0.37
POLB P06746 1/20 0.35
MAOB P27338 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7590153 0.91 TSHR (0.50) ALDH1A1LMNATSHRTDP1ESR1
SCHEMBL7595389 0.90 TSHR (0.51) ALDH1A1LMNATSHRTDP1ESR1
SCHEMBL7593446 0.88 TSHR (0.44) ALDH1A1LMNATSHRTDP1L3MBTL1
SCHEMBL7592823 0.84 ALDH1A1 (0.42) ALDH1A1LMNATSHRTDP1L3MBTL1
SCHEMBL19795490 0.82 ALDH1A1 (0.55) ALDH1A1LMNATSHRTDP1ESR1
SCHEMBL7595676 0.81 ALDH1A1 (0.49) ALDH1A1TSHRTDP1KDM4ETP53
SCHEMBL7595297 0.79 CFTR (0.50) PDK2KDM4E
SCHEMBL7591357 0.78 ALDH1A1 (0.50) ALDH1A1LMNATSHRTDP1ESR1
SCHEMBL20267555 0.78 ALDH1A1 (0.50) ALDH1A1PDK2LMNATSHRTDP1
SCHEMBL7595049 0.78 CTSS (0.33) ALDH1A1L3MBTL1KDM4EMAPK1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968994-B1 PROCESS FOR PRODUCING SUBSTITUTED TRIFLUOROBENZOIC ACIDS AND ESTERS THEREOF UBE INDUSTRIES (JP) 2002-11-06 EP claimed
EP-0968994-A1 SUBSTITUTED TRIFLUOROBENZOIC ACIDS, ESTERS THEREOF, AND PROCESS FOR PRODUCING THE SAME UBE INDUSTRIES, LTD. (JP) 2000-01-05 EP claimed
EP-0968994-B1 PROCESS FOR PRODUCING SUBSTITUTED TRIFLUOROBENZOIC ACIDS AND ESTERS THEREOF UBE INDUSTRIES (JP) 2002-11-06 EP disclosed
US-6307091-B1 TRIFLUOROMETHYLATING A TRIFLUOROIODOBENZOIC ACID ESTER WITH ADIFLUORO(FLUOROSULFONYL)ACETIC ACID ESTER IN THE PRESENCE OF A COPPER CATALYST IN AN ORGANIC SOLVENT. UBE INDUSTRIES, LTD. (JP) 2001-10-23 US disclosed
US-6160171-A Trifluoro-substituted benzoic acid, esters thereof, and process for producing the same UBE INDUSTRIES, LTD. (JP) 2000-12-12 US disclosed
EP-0968994-A1 SUBSTITUTED TRIFLUOROBENZOIC ACIDS, ESTERS THEREOF, AND PROCESS FOR PRODUCING THE SAME UBE INDUSTRIES, LTD. (JP) 2000-01-05 EP disclosed