SCHEMBL7595017

SCHEMBL7595017

Cn1c(N2CCN(CCCCC3(OC(=O)NCc4ccccc4)c4ccccc4-c4ccccc43)CC2)nc2ccccc21

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
HTR2A P28223 2/20 0.42
HTR2C P28335 2/20 0.42
HTR2B P41595 2/20 0.42
DRD2 P14416 3/20 0.41
HTR1A P08908 2/20 0.41
HTR7 P34969 1/20 0.41
DRD4 P21917 1/20 0.41
DRD3 P35462 1/20 0.41
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7596191 0.94 ALDH1A1 (0.49) ALDH1A1HTR2AHTR2CHTR2BHTR1A
SCHEMBL7601057 0.93 ALDH1A1 (0.48) ALDH1A1DRD2HTR1AHTR7
SCHEMBL7594407 0.91 ALDH1A1 (0.45) ALDH1A1HPGDSMN1; SMN2
SCHEMBL7602690 0.89 ALDH1A1 (0.44) ALDH1A1HPGDSMN1; SMN2
SCHEMBL7630436 0.87 ALDH1A1 (0.42) ALDH1A1HTR2AHTR2CHTR2BDRD2
SCHEMBL6771866 0.86 ALDH1A1 (0.58) ALDH1A1HTR2AHTR2CHTR2BDRD2
SCHEMBL7599828 0.86 ALDH1A1 (0.41) ALDH1A1HPGDSMN1; SMN2
SCHEMBL7599330 0.85 FPR3 (0.41) ALDH1A1DRD3HPGDSMN1; SMN2
SCHEMBL7603379 0.84 HTR1A (0.52) ALDH1A1HTR2AHTR2CDRD2HTR1A
SCHEMBL7608410 0.82 PKM (0.42) ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255736-A2 SUBSTITUTED PIPERAZINE DERIVATIVES AND THEIR USE AS INHIBITORS OF THE MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN (MTP) Boehringer Ingelheim Pharma KG (DE) 2002-11-13 EP disclosed
WO-2001047898-A2 SUBSTITUTED PIPERAZINE DERIVATIVES AND THEIR USE AS INHIBITORS OF THE MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN (MTP) BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-07-05 WO disclosed