Ethinyl Estradiol

Ethinyl Estradiol

SCHEMBL7602883

C#CC1(O)CCC2C3CCc4cc(O)ccc4C3CCC21C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ESR1

The experimentally established mechanism targets of Ethinyl Estradiol. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 known ✓ P03372 8/20 1.00
CYP3A4 P08684 3/20 1.00
ESR2 Q92731 3/20 1.00
NR3C1 P04150 3/20 1.00
PGR P06401 3/20 1.00
ABCB11 O95342 2/20 1.00
SLC6A2 P23975 2/20 1.00
SLC6A4 P31645 2/20 1.00
SLC6A3 Q01959 2/20 1.00
SLC22A2 O15244 1/20 1.00
NR1I2 O75469 1/20 1.00
SHBG P04278 1/20 1.00
HTR1A P08908 1/20 1.00
ADORA3 P0DMS8 1/20 1.00
AR P10275 1/20 1.00
ADRB3 P13945 1/20 1.00
CYP2B6 P20813 1/20 1.00
TBXA2R P21731 1/20 1.00
UGT1A1 P22309 1/20 1.00
PDE4A P27815 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ethinyl Estradiol SCHEMBL15213118 1.00 ESR1 (1.00) ESR1CYP3A4ESR2NR3C1PGR
Ethinyl Estradiol SCHEMBL13575761 1.00 ESR1 (1.00) ESR1CYP3A4ESR2NR3C1PGR
Ethinyl Estradiol SCHEMBL4071 1.00 ESR1 (1.00) ESR1CYP3A4ESR2NR3C1PGR
Ethinyl Estradiol SCHEMBL2389175 1.00 ESR1 (1.00) ESR1CYP3A4ESR2NR3C1PGR
Ethinyl Estradiol SCHEMBL12180049 1.00 ESR1 (1.00) ESR1CYP3A4ESR2NR3C1PGR
Ethinyl Estradiol SCHEMBL16070988 1.00 ESR1 (1.00) ESR1CYP3A4ESR2NR3C1PGR
Ethinyl Estradiol SCHEMBL5030184 1.00 ESR1 (1.00) ESR1CYP3A4ESR2NR3C1PGR
Ethinyl Estradiol SCHEMBL19963467 1.00 ESR1 (1.00) ESR1CYP3A4ESR2NR3C1PGR
Ethinyl Estradiol SCHEMBL14380029 1.00 ESR1 (1.00) ESR1CYP3A4ESR2NR3C1PGR
Ethinyl Estradiol SCHEMBL5995835 1.00 ESR1 (1.00) ESR1CYP3A4ESR2NR3C1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114720570-B Method for detecting 8 estrogens in fish meat 上海市环境科学研究院 2023-08-29 CN disclosed
CN-114720570-A Method for detecting 8 estrogens in fish 上海市环境科学研究院 2022-07-08 CN disclosed
EP-2899281-B1 Inhibitors of sterol metabolism for their use to accumulate triglycerides in microalgae, and methods thereof COMMISSARIAT ENERGIE ATOMIQUE (FR) 2020-07-01 EP disclosed
US-9107959-B2 Method for site-specific polyvalent display on polymers NEW YORK UNIVERSITY (US) 2015-08-18 US disclosed
US-9107959-B2 Method for site-specific polyvalent display on polymers NEW YORK UNIVERSITY (US) 2015-08-18 US disclosed
US-8524663-B2 Method for site-specific polyvalent display on polymers NEW YORK UNIVERSITY (US) 2013-09-03 US disclosed
US-8524663-B2 Method for site-specific polyvalent display on polymers NEW YORK UNIVERSITY (US) 2013-09-03 US disclosed
US-20120122779-A1 Method for site-specific polyvalent display on polymers NEW YORK UNIVERSITY 2012-05-17 US disclosed
US-20120122779-A1 Method for site-specific polyvalent display on polymers NEW YORK UNIVERSITY 2012-05-17 US disclosed
US-20080269425-A1 Novel Catalyst WAKO PURE CHEMICAL INDUSTRIES, LTD. (JP) 2008-10-30 US disclosed
US-20080269425-A1 Novel Catalyst WAKO PURE CHEMICAL INDUSTRIES, LTD. (JP) 2008-10-30 US disclosed
EP-1829610-A1 NOVEL CATALYST Wako Pure Chemical Industries, Ltd. (JP) 2007-09-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080269425-A1 Novel Catalyst PPOX, PNMT, POLRMT ESR1 2244/4885CYP3A4 388/4885ESR2 2822/4885
US-20120122779-A1 Method for site-specific polyvalent display on polymers NGLY1, DNPEP, GPKOW ESR1 4503/4885CYP3A4 3957/4885ESR2 4764/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.