SCHEMBL7609190

SCHEMBL7609190

c1ccn(Nc2ccncc2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 5/20 0.48
CTSD P07339 1/20 0.46
MDM2 Q00987 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
RAD52 P43351 1/20 0.37
MAP4K4 O95819 1/20 0.36
JAK2 O60674 1/20 0.35
TYK2 P29597 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626632 0.77 ALDH1A1 (0.43) SLC6A2CTSDJAK2
SCHEMBL9469956 0.76 NPC1 (0.43) RAD52MAP4K4
SCHEMBL10569077 0.73 SLC6A2 (0.46) SLC6A2CTSDMDM2TAAR1RAD52
SCHEMBL11548693 0.71 TSHR (0.46)
SCHEMBL8538989 0.70 KDR (0.37)
SCHEMBL11547917 0.70 ALDH1A1 (0.59) SLC6A2JAK2
SCHEMBL7611639 0.69 SLC6A2 (0.50) SLC6A2CTSDMAP4K4JAK2TYK2
SCHEMBL9791981 0.67 AOC1 (0.37) RAD52
SCHEMBL7608055 0.67 TGFBR1 (0.38)
Hydrochloric Acid SCHEMBL7610830 0.67 SLC6A2 (0.49) SLC6A2CTSDMAP4K4JAK2TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1184969-C Use of unsubstd and substd. N-(pyrrol-1-yl) pyridinamines as anticonvulsant agents AVENTIS PHARMA INC (US) 2005-01-19 CN claimed
EP-0840609-B1 USE OF UNSUBSTITUTED AND SUBSTITUTED N-(PYRROL-1-YL)PYRIDINAMINES AS ANTICONVULSANT AGENTS AVENTIS PHARMA INC (US) 2002-06-05 EP claimed
CN-1191486-A Use of unsubstituted and substituted N- (pyrrol-1-yl) pyridinamines as anticonvulsants HOECHST MARION ROUSSEL INC (US) 1998-08-26 CN claimed
US-5776955-A Use of unsubstituted and substituted n-(pyrrol-1-yl)pyridinamines as anticonvulsant agents HOECHST MARION ROUSSEL, INC. 1998-07-07 US claimed
EP-0840609-A1 USE OF UNSUBSTITUTED AND SUBSTITUTED N-(PYRROL-1-YL)PYRIDINAMINES AS ANTICONVULSANT AGENTS HOECHST MARION ROUSSEL, INC. (US) 1998-05-13 EP claimed
WO-1997004777-A1 USE OFF UNSUBSTITUTED AND SUBSTITUTED N-(PYRROL-1-YL)PYRIDINAMINES AS ANTICONVULSANT AGENTS HOECHST MARION ROUSSEL, INC. (US) 1997-02-13 WO claimed
US-4900742-A N-(pyrrol-1-yl)pyridinamine compounds having memory enhancing properties HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1990-02-13 US claimed
EP-0226099-A2 N-(pyrrol-1-yl)pyridinamines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1987-06-24 EP claimed
CN-1184969-C Use of unsubstd and substd. N-(pyrrol-1-yl) pyridinamines as anticonvulsant agents AVENTIS PHARMA INC (US) 2005-01-19 CN disclosed
EP-0840609-B1 USE OF UNSUBSTITUTED AND SUBSTITUTED N-(PYRROL-1-YL)PYRIDINAMINES AS ANTICONVULSANT AGENTS AVENTIS PHARMA INC (US) 2002-06-05 EP disclosed
CN-1191486-A Use of unsubstituted and substituted N- (pyrrol-1-yl) pyridinamines as anticonvulsants HOECHST MARION ROUSSEL INC (US) 1998-08-26 CN disclosed
US-5776955-A Use of unsubstituted and substituted n-(pyrrol-1-yl)pyridinamines as anticonvulsant agents HOECHST MARION ROUSSEL, INC. 1998-07-07 US disclosed
EP-0840609-A1 USE OF UNSUBSTITUTED AND SUBSTITUTED N-(PYRROL-1-YL)PYRIDINAMINES AS ANTICONVULSANT AGENTS HOECHST MARION ROUSSEL, INC. (US) 1998-05-13 EP disclosed
WO-1997004777-A1 USE OFF UNSUBSTITUTED AND SUBSTITUTED N-(PYRROL-1-YL)PYRIDINAMINES AS ANTICONVULSANT AGENTS HOECHST MARION ROUSSEL, INC. (US) 1997-02-13 WO disclosed
US-5039687-A Learning enhancement, cognition activation HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-08-13 US disclosed
US-5032599-A Learning enhancement HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-07-16 US disclosed
US-4900742-A N-(pyrrol-1-yl)pyridinamine compounds having memory enhancing properties HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1990-02-13 US disclosed
US-4792562-A N-(pyrrol-1-yl)pyridinamines having memory enhancing activity HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1988-12-20 US disclosed
US-4752610-A N-(pyrrol-1-yl)pyridinamines having memory enhancing properties HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1988-06-21 US disclosed
EP-0226099-A2 N-(pyrrol-1-yl)pyridinamines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1987-06-24 EP disclosed