SCHEMBL7651163

SCHEMBL7651163

CC(C)(C(=O)O)n1c(=O)[nH]c2cc3ccccc3cc2c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.44
FEN1 P39748 5/20 0.42
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
CA12 O43570 4/20 0.37
CA9 Q16790 4/20 0.37
NPEPPS P55786 1/20 0.37
ERCC1 P07992 2/20 0.36
ERCC4 Q92889 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7651882 0.82 ADORA3 (0.54) FEN1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL7653151 0.82 KDM4E (0.44) LMNAKDM4EALDH1A1HPGDHSD17B10
SCHEMBL7648323 0.80 SMN1; SMN2 (0.41) LMNAKDM4EALDH1A1HPGD
SCHEMBL7653637 0.80 MPO (0.43) FEN1KDM4EALDH1A1HSD17B10CA12
SCHEMBL8133826 0.79 KDM4E (0.45) LMNAFEN1KDM4EALDH1A1HPGD
SCHEMBL7650104 0.78 FEN1 (0.58) FEN1
SCHEMBL16265009 0.78 RXFP1 (0.45) LMNAALDH1A1HPGDHSD17B10
SCHEMBL7652823 0.78 CA9 (0.58) LMNAKDM4EHPGDGRIN2DGRIN3B
SCHEMBL7655193 0.78 CA12 (0.58) LMNAALDH1A1HPGDCA12CA9
SCHEMBL7650006 0.69 FEN1 (0.58) FEN1ERCC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed