SCHEMBL7652823

SCHEMBL7652823

CC(C)(C(=O)O)n1c(=O)[nH]c2cc(Cl)ccc2c1=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 3/20 0.58
CA12 O43570 2/20 0.58
KDM4E B2RXH2 2/20 0.48
HPGD P15428 2/20 0.48
GAA P10253 1/20 0.48
CMA1 P23946 1/20 0.48
LMNA P02545 3/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
CYP2C9 P11712 1/20 0.47
MAPK1 P28482 1/20 0.47
BLM P54132 1/20 0.47
TP53 P04637 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HAVCR2 Q8TDQ0 1/20 0.44
MPO P05164 1/20 0.43
XDH P47989 1/20 0.43
GRIN2D O15399 1/20 0.43
GRIN3B O60391 1/20 0.43
GRIN1 Q05586 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7655193 0.89 CA12 (0.58) CA9CA12HPGDGAALMNA
SCHEMBL31393248 0.85 CA9 (0.60) CA9CA12CMA1LMNAMEN1
SCHEMBL7648344 0.82 CA9 (0.51) CA9CA12KDM4EHPGDGAA
SCHEMBL7651882 0.80 ADORA3 (0.54) CA9CA12KDM4EHPGDGAA
SCHEMBL7649499 0.79 CA9 (0.45) CA9CA12KDM4EHPGDGAA
SCHEMBL7651163 0.78 LMNA (0.44) CA9CA12KDM4EHPGDLMNA
SCHEMBL16265009 0.78 RXFP1 (0.45) HPGDLMNAMEN1KMT2ACYP2C9
SCHEMBL7653637 0.77 MPO (0.43) CA9CA12KDM4EMPOXDH
SCHEMBL8133826 0.76 KDM4E (0.45) KDM4EHPGDGAALMNAMEN1
SCHEMBL7650104 0.75 FEN1 (0.58) MEN1KMT2AMPOXDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed