SCHEMBL7653483

SCHEMBL7653483

CCOC(=O)C(C)(C)n1c(=O)c2cc(Cl)ccc2n(CCCCBr)c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
PSEN1 P49768 5/20 0.44
PSEN2 P49810 5/20 0.44
APH1B Q8WW43 5/20 0.44
NCSTN Q92542 5/20 0.44
APH1A Q96BI3 5/20 0.44
PSENEN Q9NZ42 5/20 0.44
L3MBTL1 Q9Y468 2/20 0.42
LMNA P02545 2/20 0.42
CHEK1 O14757 2/20 0.39
KDM4E B2RXH2 2/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
CASP1 P29466 1/20 0.39
HSD17B10 Q99714 1/20 0.39
RORA P35398 1/20 0.39
RORC P51449 1/20 0.39
NR1H2 P55055 1/20 0.39
RORB Q92753 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7654685 0.92 PSEN1 (0.42) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL7651232 0.90 RORA (0.41) ALDH1A1L3MBTL1LMNAKDM4EHPGD
SCHEMBL7654237 0.88 PER2 (0.38) ALDH1A1LMNAKDM4EHTTTNF
SCHEMBL7650485 0.87 HDAC1 (0.38) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL7655134 0.85 TNF (0.51) ALDH1A1L3MBTL1LMNAKDM4EHPGD
SCHEMBL7648481 0.85 MAPT (0.46) ALDH1A1LMNA
SCHEMBL7649601 0.85 ALDH1A1 (0.37) ALDH1A1L3MBTL1LMNAKDM4ETSHR
SCHEMBL7651184 0.85 ALDH1A1 (0.50) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL7654850 0.85 ALDH1A1 (0.50) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL7653084 0.82 TNF (0.52) ALDH1A1L3MBTL1LMNAKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed