SCHEMBL7654685

SCHEMBL7654685

CCOC(=O)C(C)(C)n1c(=O)c2ccc(Cl)cc2n(CCCCBr)c1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 4/20 0.42
PSEN2 P49810 4/20 0.42
APH1B Q8WW43 4/20 0.42
NCSTN Q92542 4/20 0.42
APH1A Q96BI3 4/20 0.42
PSENEN Q9NZ42 4/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
LMNA P02545 2/20 0.42
HDAC6 Q9UBN7 3/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
ALDH1A1 P00352 6/20 0.39
TSHR P16473 3/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
ALOX15 P16050 2/20 0.39
HSD17B10 Q99714 2/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
TNF P01375 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7653483 0.92 ALDH1A1 (0.44) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7649498 0.87 HDAC6 (0.40) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7655134 0.85 TNF (0.51) L3MBTL1LMNAALDH1A1TNFKDM4E
SCHEMBL7654850 0.85 ALDH1A1 (0.50) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7651184 0.85 ALDH1A1 (0.50) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7651232 0.84 RORA (0.41) L3MBTL1LMNAALDH1A1HSD17B10TNF
SCHEMBL7653084 0.82 TNF (0.52) L3MBTL1LMNAALDH1A1TSHRHSD17B10
SCHEMBL7654237 0.82 PER2 (0.38) LMNAALDH1A1TNFKDM4EHTT
SCHEMBL7650485 0.79 HDAC1 (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7648481 0.79 MAPT (0.46) LMNAALDH1A1CYP1A2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed