SCHEMBL7654850

SCHEMBL7654850

CCOC(=O)C(C)(C)n1c(=O)c2ccccc2n(CCCCCCBr)c1=O

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
HTT P42858 1/20 0.50
TNF P01375 1/20 0.50
CNR2 P34972 7/20 0.47
KDM4E B2RXH2 6/20 0.47
LMNA P02545 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.45
MAPT P10636 1/20 0.42
PSEN1 P49768 1/20 0.41
PSEN2 P49810 1/20 0.41
APH1B Q8WW43 1/20 0.41
NCSTN Q92542 1/20 0.41
APH1A Q96BI3 1/20 0.41
PSENEN Q9NZ42 1/20 0.41
HPGD P15428 1/20 0.41
MAPK1 P28482 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7651184 1.00 ALDH1A1 (0.50) ALDH1A1HTTTNFCNR2KDM4E
SCHEMBL7655134 0.99 TNF (0.51) ALDH1A1HTTTNFCNR2KDM4E
SCHEMBL7653084 0.96 TNF (0.52) ALDH1A1HTTTNFCNR2KDM4E
SCHEMBL7652234 0.88 CNR2 (0.49) ALDH1A1HTTTNFCNR2KDM4E
SCHEMBL7651131 0.87 CNR2 (0.42) ALDH1A1HTTTNFCNR2KDM4E
SCHEMBL7651232 0.86 RORA (0.41) ALDH1A1HTTTNFCNR2KDM4E
SCHEMBL7654685 0.85 PSEN1 (0.42) ALDH1A1HTTTNFKDM4ELMNA
SCHEMBL7654237 0.85 PER2 (0.38) ALDH1A1HTTTNFCNR2KDM4E
SCHEMBL7653483 0.85 ALDH1A1 (0.44) ALDH1A1HTTTNFCNR2KDM4E
SCHEMBL7649601 0.83 ALDH1A1 (0.37) ALDH1A1HTTTNFCNR2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed