SCHEMBL7654436

SCHEMBL7654436

O=C(O)c1ccccc1CCn1c(=O)c2ccccc2n(CCCCBr)c1=O

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 5/20 0.47
HDAC6 Q9UBN7 5/20 0.47
HDAC1 Q13547 3/20 0.46
HDAC11 Q96DB2 3/20 0.46
THRB P10828 1/20 0.46
CNR2 P34972 6/20 0.45
MELK Q14680 1/20 0.44
MAPT P10636 1/20 0.43
TNF P01375 1/20 0.42
FOLH1 Q04609 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7649768 0.74 TNF (0.70) HDAC1CNR2TNF
SCHEMBL7654430 0.74 TNF (0.70) HDAC1CNR2TNF
SCHEMBL5036947 0.73 TNF (0.62) HDAC1CNR2TNF
SCHEMBL7651124 0.73 PGR (0.68) MAPT
SCHEMBL7654823 0.72 MAPT (0.52) CNR2MAPTTNF
SCHEMBL8831732 0.72 RORA (0.69) HDAC8HDAC6HDAC1HDAC11
SCHEMBL9559954 0.71 FOLH1 (0.58) FOLH1
SCHEMBL7649846 0.71 TNF (0.59) CNR2TNF
SCHEMBL8791639 0.71 FOLH1 (0.61) FOLH1
SCHEMBL6417860 0.70 CNR2 (0.68) CNR2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed