SCHEMBL7656086

SCHEMBL7656086

CN(C)CCn1c(-c2ccccc2)nn(-c2ccccc2)c1=O

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSK P43235 2/20 0.45
ADORA3 P0DMS8 4/20 0.42
ADORA2A P29274 2/20 0.41
ADORA2B P29275 2/20 0.41
POLB P06746 1/20 0.40
HPGD P15428 6/20 0.40
KDM4E B2RXH2 5/20 0.40
ALDH1A1 P00352 5/20 0.40
HSD17B10 Q99714 5/20 0.40
ALOX15 P16050 4/20 0.40
CYP3A4 P08684 3/20 0.40
TSHR P16473 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
ADORA1 P30542 1/20 0.39
ROCK2 O75116 1/20 0.39
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7652516 0.92 CTSK (0.46) CTSKPOLBHPGDKDM4EALDH1A1
SCHEMBL7652922 0.90 CTSK (0.50) CTSKADORA3ADORA2AALDH1A1MEN1
SCHEMBL7679154 0.89 ALDH1A1 (0.46) CTSKADORA3POLBKDM4EALDH1A1
SCHEMBL7649212 0.89 CTSK (0.47) CTSKADORA2APOLBHPGDKDM4E
SCHEMBL7652478 0.88 CTSK (0.48) CTSKADORA3ADORA2AADORA1ROCK2
SCHEMBL7652889 0.87 CTSK (0.45) CTSKADORA3ADORA2AKDM4EALDH1A1
SCHEMBL7656565 0.86 ROCK2 (0.48) CTSKADORA3ADORA2APOLBALDH1A1
SCHEMBL7655384 0.85 HPGD (0.43) ADORA3ADORA2AADORA2BPOLBHPGD
SCHEMBL7652938 0.85 ALDH1A1 (0.43) CTSKADORA3ADORA2AADORA2BHPGD
SCHEMBL7656105 0.84 DRD2 (0.39) CTSKADORA3ADORA2AADORA2BHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492407-B2 NEUROPROTECTIVE ACTIVITY BOEHRINGER IMGELHEIM PHARMA KG (DE) 2002-12-10 US disclosed