SCHEMBL7659173

SCHEMBL7659173

Cc1c(NC(=O)c2ccco2)ccc2oc(N[C@@H](Cc3ccccc3)C(=O)O)nc(=O)c12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.43
KMT2A Q03164 6/20 0.42
MEN1 O00255 5/20 0.42
RAB9A P51151 4/20 0.42
MAPT P10636 3/20 0.42
NPC1 O15118 3/20 0.42
HPGD P15428 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
ELANE P08246 2/20 0.41
TSHR P16473 1/20 0.40
ALDH1A1 P00352 1/20 0.40
KDM4E B2RXH2 2/20 0.40
CTSL P07711 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6507056 0.86 CTRB1 (0.51) ATMKMT2AMEN1RAB9AMAPT
SCHEMBL8549217 0.84 ELANE (0.41) ATMKMT2AMEN1MAPTHPGD
SCHEMBL8545041 0.84 ELANE (0.43) KMT2AMEN1ELANEALDH1A1PPARG
SCHEMBL8550797 0.81 ALDH1A1 (0.42) KMT2AMEN1RAB9AMAPTNPC1
SCHEMBL8545895 0.77 ALDH1A1 (0.50) KMT2AMEN1ELANETSHRALDH1A1
SCHEMBL8549764 0.77 ELANE (0.47) KMT2AMEN1ELANEALDH1A1PPARG
SCHEMBL6497371 0.72 NPC1 (0.47) KMT2AMEN1RAB9AMAPTNPC1
SCHEMBL6496066 0.72 CTRB1 (0.67) ATMKMT2AMEN1RAB9AMAPT
SCHEMBL7813812 0.71 CTRB1 (0.52) KMT2AMEN1RAB9ANPC1HPGD
SCHEMBL6499604 0.71 CTRB1 (0.56) KMT2AMEN1SMN1; SMN2ELANEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6380189-B1 FOR TREATING HERPES-RELATED DISORDERS G.D. SEARLE & CO. 2002-04-30 US disclosed
EP-0828721-A1 2-AMINO-BENZOXAZINONES FOR THE TREATMENT OF VIRAL INFECTIONS G.D. SEARLE & CO. (US) 1998-03-18 EP disclosed