SCHEMBL7663166

SCHEMBL7663166

O=C(OCc1ccccc1)[C@@H]1CCCCN1c1nc2cc(Cl)ccc2o1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGES O14684 14/20 0.53
PTGS2 P35354 5/20 0.53
FKBP1A P62942 3/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
HCRTR1 O43613 1/20 0.44
HCRTR2 O43614 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7664466 0.90 FKBP1A (0.48) PTGESPTGS2FKBP1ANPC1RAB9A
SCHEMBL27559144 0.86 ALDH1A1 (0.44) PTGESPTGS2FKBP1ANPC1RAB9A
SCHEMBL7826244 0.86 FKBP1A (0.48) FKBP1ANPC1RAB9A
SCHEMBL6737810 0.83 PTGES (0.56) PTGESPTGS2HCRTR1HCRTR2
SCHEMBL8027454 0.80 FKBP1A (0.45) FKBP1ANPC1RAB9A
SCHEMBL6740429 0.80 PTGES (0.54) PTGESPTGS2
SCHEMBL7655863 0.75 GABRP (0.45) NPC1RAB9AHCRTR1HCRTR2
SCHEMBL6739627 0.75 LMNA (0.52) FKBP1A
SCHEMBL23018138 0.73 XDH (0.58) PTGESPTGS2
SCHEMBL27479845 0.73 LMNA (0.51) NPC1RAB9AHCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6495549-B1 1-HETEROARYL-PIPERIDINE DERIVATIVES; MODERATING NEURONAL DEGENERATION; PROMOTING NEURONAL REGENERATION AND OUTGROWTH; TREATOG NEUROLOGICAL DISORDERS ARISING FROM NEURODEGENERATIVE DISEASES OR OTHER DISORDERS INVOLVING NERVE DAMAGE PFIZER INC 2002-12-17 US disclosed
CN-1315951-A FKBP inhibitors PFIZER LTD (US) 2001-10-03 CN disclosed