SCHEMBL7667709

SCHEMBL7667709

COC(=O)c1cc(CNC(Cn2ccnc2)c2ccc(F)cc2)ccc1Cc1ccc(F)cc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.39
KDM4E B2RXH2 2/20 0.38
TBXAS1 P24557 1/20 0.38
AHR P35869 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
LMNA P02545 1/20 0.38
CYP19A1 P11511 3/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
CYP51A1 Q16850 2/20 0.37
IDO1 P14902 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7664949 0.91 PTGS2 (0.40) PTGS2LMNACYP19A1CYP11B1CYP11B2
SCHEMBL7667718 0.83 CYP19A1 (0.40) PTGS2KDM4ETBXAS1AHRNPSR1
SCHEMBL7667706 0.83 TBXAS1 (0.41) PTGS2KDM4ETBXAS1AHRNPSR1
SCHEMBL7653717 0.81 FNTA (0.51) NPSR1
SCHEMBL7665403 0.76 CYP19A1 (0.41) PTGS2CYP19A1CYP11B1CYP11B2CYP51A1
SCHEMBL7653706 0.75 PTGS2 (0.47) PTGS2KDM4EAHRNPSR1CYP51A1
SCHEMBL7657859 0.74 FNTA (0.51) NPSR1
SCHEMBL7662187 0.73 FNTA (0.52) PTGS2CYP51A1CYP3A4CYP2D6CYP2C9
SCHEMBL7662191 0.72 FNTA (0.38) PTGS2LMNACYP51A1CYP3A4CYP2D6
SCHEMBL7664955 0.72 CYP19A1 (0.45) TBXAS1LMNACYP19A1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6410539-B1 ANTICARCINOGENIC AGENTS ASTRAZENCA UK LIMITED (GB) 2002-06-25 US disclosed