SCHEMBL7670109

SCHEMBL7670109

O=C(O)N(CBr)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.49
GSK3B P49841 2/20 0.49
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
RORC P51449 1/20 0.42
SRD5A2 P31213 2/20 0.42
MLYCD O95822 4/20 0.40
SERPINE1 P05121 2/20 0.40
MTOR P42345 1/20 0.39
PDK2 Q15119 1/20 0.39
PDK4 Q16654 1/20 0.39
EPHX2 P34913 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044376 0.84 CES2 (0.44) PTPN1GSK3BCES2CES1RORC
SCHEMBL6229257 0.82 MLYCD (0.54) CES2CES1MLYCDSERPINE1MTOR
SCHEMBL7669043 0.78 PTPN1 (0.41) PTPN1GSK3BCES2CES1MLYCD
SCHEMBL13735234 0.77 ALDH1A1 (0.52) PTPN1GSK3B
SCHEMBL28102660 0.73 CES2 (0.48) PTPN1GSK3BCES2CES1SRD5A2
SCHEMBL1978108 0.72 CES2 (0.47) PTPN1GSK3BCES2CES1SRD5A2
SCHEMBL2094862 0.72 SMN1; SMN2 (0.51) CES2CES1SRD5A2MLYCDMTOR
SCHEMBL3065041 0.70 TSHR (0.56) RORCMLYCDMTORPDK2PDK4
SCHEMBL18360376 0.70 KEAP1 (0.46) PTPN1GSK3BCES2CES1SRD5A2
SCHEMBL2097683 0.70 NPSR1 (0.48) CES2CES1SRD5A2MTOREPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6369221-B1 Thiazolobenzoheterocycles, preparation and medicines containing same AVENTIS PHARMA S.A. (FR) 2002-04-09 US disclosed