SCHEMBL7673680

SCHEMBL7673680

C=CCC(C#N)(CC=C)c1cccc(OC)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.40
PDE4A P27815 2/20 0.39
PDE4B Q07343 2/20 0.39
PDE4C Q08493 2/20 0.39
PDE4D Q08499 2/20 0.39
CASP1 P29466 1/20 0.38
HSD17B10 Q99714 1/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
MAPK1 P28482 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ALDH1A1 P00352 3/20 0.37
ALOX12 P18054 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ACHE P22303 1/20 0.37
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
PGR P06401 1/20 0.36
AR P10275 1/20 0.36
CA1 P00915 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9079258 0.93 KIF11 (0.37) KIF11PDE4APDE4BPDE4CPDE4D
SCHEMBL9079230 0.83 KIF11 (0.42) KIF11PDE4APDE4BPDE4CPDE4D
SCHEMBL4430846 0.80 TP53 (0.39) KIF11CASP1HSD17B10NPC1SMN1; SMN2
SCHEMBL4874767 0.79 CASP1 (0.44) KIF11PDE4APDE4BPDE4CPDE4D
SCHEMBL1007659 0.77 ACHE (0.44) KIF11PDE4APDE4BPDE4CPDE4D
SCHEMBL9080465 0.76 ALDH1A1 (0.38) KIF11HSD17B10ALDH1A1ACHEAR
SCHEMBL10624241 0.75 ALDH1A1 (0.48) RAB9ASMN1; SMN2ALDH1A1NPSR1CYP3A4
SCHEMBL9080579 0.74 MAOB (0.43) KIF11USP2IDO1AGXT
SCHEMBL11074467 0.74 LMNA (0.46) KIF11CASP1HSD17B10NPC1RAB9A
SCHEMBL6821384 0.74 TAAR1 (0.43) IDO1AGXT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6444679-B1 NEUROLOGICAL AND GASTROINTESTINAL DISORDERS; DELTA OPIOID LIGANDS OR OPIOID RECEPTORS PFIZER INC 2002-09-03 US disclosed
EP-1038872-A1 4-Phenyl-4-heteroarylpiperdine derivatives as opioid receptor ligands Pfizer Products Inc. (US) 2000-09-27 EP disclosed
US-5519022-A α, α dialkylbenzyl derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1996-05-21 US disclosed
US-5288742-A Lipoxygenase inhibitor IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-02-22 US disclosed
EP-0505122-A1 Alpha, alpha-dialkylbenzyl derivatives ZENECA LIMITED (GB) 1992-09-23 EP disclosed