SCHEMBL7677748

SCHEMBL7677748

Cn1cnnc1SCCCCCN1CCN(c2cccc(C(F)(F)F)c2)CC1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.54
HTR7 P34969 8/20 0.54
DRD2 P14416 6/20 0.50
DRD3 P35462 3/20 0.50
ADRA1A P35348 2/20 0.50
DRD5 P21918 1/20 0.50
HTR1A P08908 2/20 0.49
HTR2A P28223 2/20 0.49
HTR6 P50406 2/20 0.49
HRH4 Q9H3N8 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7680682 0.96 SIGMAR1 (0.53) SIGMAR1HTR7DRD2DRD3ADRA1A
SCHEMBL7674560 0.81 DRD2 (0.62) SIGMAR1HTR7DRD2DRD3ADRA1A
SCHEMBL12468732 0.80 DRD2 (0.54) SIGMAR1HTR7DRD2DRD3ADRA1A
SCHEMBL7677755 0.79 SIGMAR1 (0.55) SIGMAR1HTR7DRD2DRD3ADRA1A
SCHEMBL4608504 0.79 HTR7 (0.53) SIGMAR1HTR7DRD2DRD3ADRA1A
SCHEMBL12469317 0.78 NPSR1 (0.61) SIGMAR1HTR7DRD2DRD3ADRA1A
SCHEMBL7047855 0.78 DRD2 (0.64) SIGMAR1HTR7DRD2DRD3ADRA1A
SCHEMBL4608940 0.77 ALDH1A1 (0.53) SIGMAR1HTR7DRD2DRD3ADRA1A
SCHEMBL11465528 0.77 SIGMAR1 (0.76) SIGMAR1HTR7DRD2DRD3ADRA1A
SCHEMBL13875122 0.76 SIGMAR1 (0.71) SIGMAR1HTR7DRD2DRD3ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403593-B1 DOPAMINE RECEPTOR ABBOTT LABORATORIES 2002-06-11 US disclosed
US-6124294-A COMPOUNDS HAVING HIGH AFFINITY FOR DOPAMINE D3 RECEPTOR; USED TO TREAT DISORDERS WHICH RESPOND TO DOPAMINE D3 LIGANDS BASF AKTIENGESELLSCHAFT (DE) 2000-09-26 US disclosed
EP-0772604-B1 TRIAZOLE COMPOUNDS AND THEIR USE AS DOPAMINE-D3-LIGANDS BASF AG (DE) 1999-05-06 EP disclosed