SCHEMBL7679913

SCHEMBL7679913

CCOC(=O)c1cnc(NCCc2ccccn2)cc1-c1ccco1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 18/20 0.44
ADORA2A P29274 18/20 0.44
ADORA1 P30542 18/20 0.44
ADORA2B P29275 8/20 0.44
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
MAPT P10636 2/20 0.44
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5093408 0.82 ADORA3 (0.47) ADORA3ADORA2AADORA1ADORA2BKDM4E
SCHEMBL7146465 0.74 PDE4A (0.41) ADORA3ADORA2AADORA1ADORA2BKDM4E
SCHEMBL31141656 0.71 MAPT (0.53) KDM4EALDH1A1MAPT
SCHEMBL27559848 0.69 PKM (0.44) ADORA3ADORA2AADORA1ADORA2BKDM4E
SCHEMBL14255689 0.69 TSHR (0.59) ADORA3ADORA2AADORA1ADORA2BKDM4E
SCHEMBL5264243 0.68 ALDH1A1 (0.48) KDM4EALDH1A1MAPTNPSR1
SCHEMBL5089195 0.68 ALDH1A1 (0.48) ADORA1KDM4EALDH1A1MAPTNPSR1
SCHEMBL4183360 0.68 ALDH1A1 (0.48) KDM4EALDH1A1MAPTNPSR1
SCHEMBL5093430 0.67 RAB9A (0.49) KDM4EALDH1A1MAPTNPSR1
SCHEMBL1108633 0.67 CYP1A2 (0.69) KDM4EALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6417185-B1 HETEROCYCLIC ENZYME INHIBITORS CHIRON CORPORATION 2002-07-09 US disclosed