SCHEMBL7682555

SCHEMBL7682555

CC(c1ccccc1)N1CCN(C(=O)NC2CCCCC2)[C@@H](C(=O)NCCc2cnc(Cc3ccc(C#N)cc3)[nH]2)C1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 2/20 0.40
FNTA P49354 5/20 0.39
FNTB P49356 5/20 0.39
PRKAA2 P54646 3/20 0.37
GPBAR1 Q8TDU6 3/20 0.37
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.35
ERG P11308 1/20 0.35
HAT1 O14929 2/20 0.35
EP300 Q09472 2/20 0.35
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
BRS3 P32247 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6180669 0.83 FNTA (0.46) FNTAFNTB
SCHEMBL6215244 0.74 FNTA (0.40) FNTAFNTBALDH1A1
SCHEMBL7841490 0.72 CHRM4 (0.54) GPBAR1ERGEP300BRS3
Hydrochloric Acid SCHEMBL7845666 0.71 CHRM4 (0.53) GPBAR1ERGEP300BRS3
SCHEMBL7459728 0.70 FNTA (0.42) FNTAFNTBPRKAA2GPBAR1CYP3A4
Hydrochloric Acid SCHEMBL7452346 0.70 FNTA (0.42) FNTAFNTBPRKAA2GPBAR1CYP3A4
SCHEMBL6178566 0.68 FNTA (0.42) FNTAFNTBALDH1A1CYP3A4CNR1
SCHEMBL7679202 0.68 FNTA (0.48) FNTAFNTBPRKAA2ALDH1A1
SCHEMBL6179814 0.67 FNTA (0.46) FNTAFNTB
SCHEMBL2226022 0.67 FNTA (0.44) FNTAFNTBALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6432959-B1 ANTITUMOR AGENTS SCHERING CORPORATION 2002-08-13 US disclosed