SCHEMBL7683547

SCHEMBL7683547

COc1ccccc1C1CC(=O)c2c(C)n[nH]c2C1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAP1LC3B Q9GZQ8 2/20 0.50
ADRA1A P35348 2/20 0.44
ADRA1D P25100 1/20 0.44
HTR2C P28335 2/20 0.43
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42
PKM P14618 1/20 0.41
GSK3B P49841 3/20 0.40
GSK3A P49840 2/20 0.40
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TP53 P04637 1/20 0.39
CDK5 Q00535 1/20 0.39
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
KMT2A Q03164 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
CYP19A1 P11511 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7689241 0.84 HCAR2 (0.48) MAP1LC3BHTR2CLMNATSHRPKM
SCHEMBL7682852 0.82 HSD17B10 (0.39) LMNATSHRPKMHTTTP53
SCHEMBL7683237 0.82 SMN1; SMN2 (0.48) MAP1LC3BADRA1ALMNATSHRPKM
Hydrochloric Acid SCHEMBL7686909 0.74 ADRA1D (0.36) MAP1LC3BADRA1AADRA1DHTR2CLMNA
SCHEMBL1779006 0.73 HSP90AA1 (0.66) MAP1LC3BLMNATSHRPKMHTT
SCHEMBL7683944 0.72 MAP1LC3B (0.53) MAP1LC3BADRA1AADRA1D
SCHEMBL7689368 0.72 PIM1 (0.45) MAP1LC3BLMNATSHRPKMHTT
Hydrochloric Acid SCHEMBL7687660 0.72 PIM1 (0.44) MAP1LC3BLMNATSHRPKMHTT
SCHEMBL7680888 0.71 MAP1LC3B (0.51) MAP1LC3BHTR2CLMNAPKMMEN1
SCHEMBL6922001 0.70 PKM (0.58) MAP1LC3BADRA1AADRA1DHTR2CLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6350749-B1 SODIUM CHANNEL MODULATORS, ANTIARRHYTHMIA AND HYPOTENSIVE AGENTS; CARDIOVASCULAR DISORDERS, ANGINA PECTORIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-02-26 US disclosed
EP-1057812-A1 AMINOGUANIDINE HYDRAZONE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND DRUGS THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-12-06 EP disclosed