SCHEMBL7686665

SCHEMBL7686665

Cn1cnc2c1C(c1ccc(C#N)c(F)c1)N(C(=O)CCNS(=O)(=O)c1cccc(O)c1)CC2

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 13/20 0.39
TRPV4 Q9HBA0 2/20 0.35
TPH1 P17752 1/20 0.33
LMNA P02545 3/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ALDH1A1 P00352 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7681015 0.91 L3MBTL1 (0.39) KIF11TRPV4TPH1MAPTALDH1A1
SCHEMBL7680485 0.66 GPR119 (0.43) TPH1MAPTALDH1A1
SCHEMBL7680493 0.64 GPR119 (0.42) TPH1MAPTALDH1A1
SCHEMBL7228470 0.64 TRPV4 (0.35) TRPV4MAPT
SCHEMBL7686709 0.63 CYP11B1 (0.36)
Trifluoroacetic Acid SCHEMBL7227919 0.61 FNTA (0.34) TRPV4
SCHEMBL3569646 0.61 KIF11 (0.81) KIF11MAPT
SCHEMBL20743638 0.59 PKM (0.54) TRPV4MAPTALDH1A1
SCHEMBL30309628 0.59 PKM (0.54) TRPV4MAPTALDH1A1
SCHEMBL7220418 0.59 ALDH1A1 (0.40) TRPV4LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6350755-B1 PEPTIDOMIMETIC COMPOUNDS THAT DO NOT HAVE A THIOL MOIETY; THERAPY OF ARTERIOSCLEROSIS AND DIABETIC VASCULAR PATHOLOGIES; MERCK & CO., INC. 2002-02-26 US disclosed
WO-2001051128-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-07-19 WO disclosed