SCHEMBL7694103

SCHEMBL7694103

CSc1nc(C(F)(F)F)cc(=O)n1-c1cc(F)c(C#N)cc1F

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 2/20 0.40
BCAT2 O15382 7/20 0.38
BCAT1 P54687 7/20 0.38
POLB P06746 1/20 0.37
GAA P10253 1/20 0.37
PKM P14618 1/20 0.35
LMNA P02545 1/20 0.34
NPSR1 Q6W5P4 1/20 0.33
ALPL P05186 1/20 0.33
ALPI P09923 1/20 0.33
TRPV4 Q9HBA0 1/20 0.33
TSHR P16473 1/20 0.33
PDE7A Q13946 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7082848 0.81 BCAT2 (0.38) MEN1KMT2AALDH1A1BCAT2BCAT1
SCHEMBL8193399 0.79 ALPL (0.39) ALDH1A1BCAT2BCAT1ALPLALPI
SCHEMBL8129698 0.79 PDE7A (0.47) MEN1KMT2AALDH1A1POLBGAA
SCHEMBL7085889 0.72 TRPV4 (0.37) ALDH1A1BCAT2BCAT1ALPLALPI
SCHEMBL7692441 0.71 BCAT2 (0.39) BCAT2BCAT1TRPV4
SCHEMBL8193759 0.71 BCAT2 (0.40) BCAT2BCAT1TRPV4
SCHEMBL5922790 0.69 BCAT1 (0.67) BCAT2BCAT1
SCHEMBL7499656 0.69 BCAT2 (0.41) BCAT2BCAT1TRPV4
SCHEMBL8927953 0.68 BCAT2 (0.40) BCAT2BCAT1TRPV4
SCHEMBL8190553 0.68 AR (0.42) ALDH1A1BCAT2BCAT1LMNATRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6339044-B1 USEFUL AS HERBICIDES AND INSECTICIDES BAYER AKTIENGESELLSCHAFT 2002-01-15 US disclosed
EP-0736014-A1 N-CYANOARYL NITROGEN HETEROCYCLES WITH SULPHUR-CONTAINING GROUPINGS BAYER AG (DE) 1996-10-09 EP disclosed
WO-1995017391-A1 N-CYANOARYL NITROGEN HETEROCYCLES WITH SULPHUR-CONTAINING GROUPINGS BAYER AKTIENGESELLSCHAFT (DE) 1995-06-29 WO disclosed