SCHEMBL7696161

SCHEMBL7696161

C=C(c1ccc2ccccc2c1)c1ccccc1C(=O)N[C@@H](Cc1ccccc1)C(=O)CNC(C)=O

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSB P07858 4/20 0.43
CTSL P07711 3/20 0.43
CAPN1 P07384 3/20 0.43
CTSS P25774 3/20 0.43
CTSK P43235 2/20 0.43
CASP1 P29466 1/20 0.42
PIN1 Q13526 4/20 0.41
ACE P12821 2/20 0.40
CA2 P00918 1/20 0.40
CCKAR P32238 1/20 0.39
CCKBR P32239 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CCR1 P32246 1/20 0.38
CTSV O60911 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7693478 0.91 ACE (0.45) CTSBCTSLCAPN1CTSSCTSK
SCHEMBL7694857 0.87 CA2 (0.43) CTSBCTSLCAPN1CTSSCTSK
SCHEMBL7701518 0.84 CA2 (0.44) CTSBCTSLCAPN1CASP1PIN1
SCHEMBL7695603 0.79 CAPN1 (0.70) CTSBCTSLCAPN1CTSSCTSK
SCHEMBL7694848 0.78 PTPN1 (0.55) CTSBCTSLCAPN1CTSSCTSK
SCHEMBL7696723 0.77 CTSS (0.50) CTSBCTSLCTSSCTSKCASP1
SCHEMBL7698402 0.77 CHRNB2 (0.52) CTSBCTSLCAPN1CTSSCTSK
SCHEMBL7689558 0.76 ALDH1A1 (0.55) CTSBCTSLCTSSCTSKCA2
SCHEMBL7694696 0.75 KDM4E (0.47) CTSSCTSKL3MBTL1
SCHEMBL7695396 0.72 AKR1C3 (0.48) CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436925-B1 BETTER ABLE TO CROSS MEMBRANES; INHIBITORS OF CYSTEINE PROTEASES LIKE CALPAIN I AND II AND CATHEPSIN B AND L, CAN THUS BE USED TO CONTROL DISEASES ASSOCIATED WITH AN ELEVATED ACTIVITY OF CALPAIN ENZYMES OR CATHEPSIN ENZYMES ABBOTT LABORATORIES 2002-08-20 US disclosed