SCHEMBL7701518

SCHEMBL7701518

C=C(c1ccc2ccccc2c1)c1ccccc1C(=O)N[C@@H](Cc1ccccc1)C(=O)CNS(=O)(=O)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.44
KAT6A Q92794 1/20 0.44
KCNA5 P22460 3/20 0.43
CASP1 P29466 1/20 0.43
CAPN1 P07384 2/20 0.41
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
PLAT P00750 2/20 0.40
CA1 P00915 1/20 0.40
F2 P00734 1/20 0.40
PIN1 Q13526 3/20 0.39
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
ITGB1 P05556 1/20 0.39
ITGA4 P13612 1/20 0.39
PLAU P00749 1/20 0.39
NPY5R Q15761 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7694857 0.90 CA2 (0.43) CA2KAT6AKCNA5CASP1CAPN1
SCHEMBL7693478 0.85 ACE (0.45) CA2CASP1CAPN1CTSLCTSB
SCHEMBL7696161 0.84 CTSB (0.43) CA2CASP1CAPN1CTSLCTSB
SCHEMBL7700700 0.81 CA2 (0.52) CA2KAT6ACASP1CTSLCTSB
SCHEMBL7698802 0.80 CAPN1 (0.67) CA2KAT6AKCNA5CASP1CAPN1
SCHEMBL7702126 0.80 PLAT (0.45) CA2KAT6AKCNA5CASP1PLAT
SCHEMBL7703565 0.80 CA2 (0.51) CA2KAT6APLATCA1F2
SCHEMBL7701695 0.79 CA2 (0.52) CA2CASP1ITGB1ITGA4
SCHEMBL7704769 0.78 CA2 (0.52) CA2KAT6ACASP1CTSLCTSB
SCHEMBL7704469 0.78 KCNA5 (0.52) CA2KAT6AKCNA5CASP1CAPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436925-B1 BETTER ABLE TO CROSS MEMBRANES; INHIBITORS OF CYSTEINE PROTEASES LIKE CALPAIN I AND II AND CATHEPSIN B AND L, CAN THUS BE USED TO CONTROL DISEASES ASSOCIATED WITH AN ELEVATED ACTIVITY OF CALPAIN ENZYMES OR CATHEPSIN ENZYMES ABBOTT LABORATORIES 2002-08-20 US disclosed