SCHEMBL7702747

SCHEMBL7702747

N=C(N)c1ccc(C(N)=O)cn1.O=C(O)[C@@H]1CCCN1C(=O)[C@H]1NCCC1c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 8/20 0.39
OPRM1 P35372 1/20 0.38
OPRK1 P41145 1/20 0.38
ACE P12821 1/20 0.36
PRSS1 P07477 1/20 0.35
TMPRSS15 P98073 1/20 0.35
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CA2 P00918 1/20 0.35
F2 P00734 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6484948 0.82 DPP4 (0.40) DGAT1ALDH1A1CA2
SCHEMBL8723763 0.74 PRSS1 (0.42) DGAT1ACEPRSS1TMPRSS15ALDH1A1
SCHEMBL8933085 0.72 HSD11B1 (0.40) DGAT1ACEPRSS1TMPRSS15ALDH1A1
Proline SCHEMBL8727242 0.70 NOS2 (0.39) OPRK1SMN1; SMN2F2
SCHEMBL6476423 0.70 F2 (0.47) ALDH1A1SMN1; SMN2F2
SCHEMBL8722619 0.70 F2 (0.40) DGAT1OPRM1OPRK1F2
SCHEMBL6484032 0.70 PRSS1 (0.38) DGAT1PRSS1TMPRSS15ALDH1A1CA2
SCHEMBL7705659 0.68 F2 (0.33) DGAT1OPRM1PRSS1TMPRSS15ALDH1A1
SCHEMBL6476554 0.66 NNMT (0.57) SMN1; SMN2
SCHEMBL8725887 0.66 F2 (0.40) OPRM1OPRK1PRSS1F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6444817-B1 ANTICOAGULANTS ABBOTT LABORATORIES 2002-09-03 US disclosed
US-6030972-A 2- OR 5-AMINOMETHYL,2- OR 5-CYANOPYRIMIDINES AS INTERMEDIATES OF ANTICOAGULANTS IN EXTRACORPOREAL CIRCULATION (HEART-LUNG MACHINE, HEMODIALYSIS) BASF AKTIENGESELLSCHAFT (DE) 2000-02-29 US disclosed
EP-0873356-A1 NOVEL DIPEPTIDE AMIDINES AS THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1998-10-28 EP disclosed
WO-1996025426-A9 NOVEL DIPEPTIDE AMIDINES AS THROMBIN INHIBITORS 1997-06-12 WO disclosed
WO-1996025426-A1 NOVEL DIPEPTIDE AMIDINES AS THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1996-08-22 WO disclosed