SCHEMBL7703689

SCHEMBL7703689

CC(C)(C)ON1C(=O)c2ccc(N3CCCC3)c3cc([N+](=O)[O-])cc(c23)C1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.41
CYP1A2 P05177 3/20 0.41
CYP3A4 P08684 3/20 0.41
CYP2C19 P33261 3/20 0.41
CYP2C9 P11712 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
GAA P10253 2/20 0.41
SMN1; SMN2 Q16637 7/20 0.40
HTT P42858 2/20 0.40
CYP2D6 P10635 1/20 0.40
MCOLN3 Q8TDD5 1/20 0.40
LMNA P02545 5/20 0.39
MAPT P10636 4/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
RAB9A P51151 2/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
PABPC1 P11940 1/20 0.39
S1PR1 P21453 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7703730 0.83 ALDH1A1 (0.36) ALDH1A1CYP1A2CYP3A4CYP2C19CYP2C9
SCHEMBL7709865 0.82 ALDH1A1 (0.37) ALDH1A1CYP1A2SMN1; SMN2LMNAMAPT
SCHEMBL7706867 0.82 MEN1 (0.47) ALDH1A1CYP1A2CYP3A4CYP2C19CYP2C9
SCHEMBL7709480 0.77 ALDH1A1 (0.62) ALDH1A1CYP1A2CYP2C19CYP2C9NPSR1
SCHEMBL7703748 0.76 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2HTTLMNAMAPT
SCHEMBL7703715 0.73 TERT (0.37) ALDH1A1NPSR1GAAHTTMAPT
SCHEMBL4876279 0.70 GAA (0.62) ALDH1A1CYP1A2CYP2C19CYP2C9GAA
SCHEMBL7703729 0.68 MEN1 (0.44) ALDH1A1CYP1A2CYP3A4CYP2C19CYP2C9
SCHEMBL7703381 0.66 BCHE (0.39) ALDH1A1CYP1A2CYP3A4CYP2C19CYP2C9
SCHEMBL7703797 0.65 ALDH1A1 (0.44) ALDH1A1NPSR1GAASMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US disclosed
US-6177423-B1 N-(HYDROXY OR PROTECTED HYDROXY)-BENZO(DE)ISOQUINOLINE-1,3-DIONE DERIVATIVES; BACTERIAL DNA GYRASE AND DNA TOPOISOMERASE INHIBITORS USEFUL FOR ANTIBACTERIAL AGENTS HAVING REDUCED DRUG RESISTANCE AND REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed
EP-0939754-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1999-09-08 EP disclosed
WO-1998019648-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed