SCHEMBL7704047

SCHEMBL7704047

c1ccc2c(c1)CCN=C2c1ccc(N2CCOCC2)nc1

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 11/20 0.65
TDO2 P48775 1/20 0.42
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
HSD17B10 Q99714 1/20 0.42
BRD4 O60885 1/20 0.41
CREBBP Q92793 1/20 0.41
ADRA1A P35348 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7704878 0.86 CNR2 (0.47) CNR2TDO2BRD4CREBBP
SCHEMBL3249571 0.79 CNR2 (1.00) CNR2TDO2
SCHEMBL7699664 0.75 HRH3 (0.55) CNR2ALDH1A1LMNA
SCHEMBL16773016 0.74 CNR2 (0.69) CNR2ALDH1A1KDM4ELMNAMAPT
SCHEMBL7702344 0.73 MAOA (0.47)
SCHEMBL7702043 0.73 NOS3 (0.44) ALDH1A1KDM4ELMNA
SCHEMBL7705693 0.72 NOS3 (0.42) TDO2ALDH1A1KDM4ELMNA
SCHEMBL3239421 0.71 CNR2 (0.66) CNR2TDO2ALDH1A1KDM4EHPGD
SCHEMBL3648791 0.71 CNR2 (0.66) CNR2TDO2BRD4CREBBP
SCHEMBL7697815 0.70 NOS3 (0.41) ALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901488-B1 2,4-DIAMINOPYRIMIDINE DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2002-11-06 EP disclosed
EP-0901488-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-17 EP disclosed
US-5866583-A Substituted 2,4-diaminopyrimidines HOFFMANN-LA ROCHE INC. (US) 1999-02-02 US disclosed
WO-1997043277-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-11-20 WO disclosed