SCHEMBL7705872

SCHEMBL7705872

COc1ccnc(C2=NCCc3ccccc32)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.52
CCR1 P32246 1/20 0.51
CCR5 P51681 1/20 0.51
CCR8 P51685 1/20 0.51
PKM P14618 1/20 0.44
RAD52 P43351 1/20 0.44
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
MAPK10 P53779 4/20 0.43
LMNA P02545 2/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
NOS3 P29474 1/20 0.41
NOS2 P35228 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7702378 0.81 NPY5R (0.54) MAOAPKMRAD52CA1CA2
SCHEMBL28338943 0.79 HTR7 (0.55) MAOACA1CA2CA7CA9
SCHEMBL7704052 0.79 GRIN2D (0.45) MAOAPKMRAD52MAPK10LMNA
SCHEMBL7705661 0.78 NOS3 (0.44) MAOACCR1CCR5CCR8MAPK10
SCHEMBL7701012 0.77 NOS3 (0.49) MAOACCR1CCR5CCR8PKM
SCHEMBL12567716 0.77 ALDH1A1 (0.65) MAOAPKMRAD52CA1CA2
SCHEMBL29498350 0.77 ALDH1A1 (0.65) MAOAPKMRAD52CA1CA2
SCHEMBL29498357 0.77 ALDH1A1 (0.65) MAOAPKMRAD52CA1CA2
SCHEMBL27909626 0.76 CCR1 (0.61) CCR1CCR5CCR8LMNAALDH1A1
SCHEMBL7705613 0.74 NOS3 (0.45) MAOAALDH1A1NOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901488-B1 2,4-DIAMINOPYRIMIDINE DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2002-11-06 EP disclosed
EP-0901488-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-17 EP disclosed
US-5866583-A Substituted 2,4-diaminopyrimidines HOFFMANN-LA ROCHE INC. (US) 1999-02-02 US disclosed
WO-1997043277-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-11-20 WO disclosed