SCHEMBL7707715

SCHEMBL7707715

CCC(=O)c1c(C(C)=O)c2ccc(C(=O)O)cc2n1Cc1cc2c(cc1Cl)OCO2

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 1/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
EDNRA P25101 14/20 0.42
EDNRB P24530 11/20 0.42
MAPK8 P45983 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPK1 P28482 1/20 0.38
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7424082 0.85 SLC22A12 (0.42) SLC22A12CA12CA1CA2CA9
SCHEMBL7422706 0.78 SLC22A12 (0.41) SLC22A12EDNRAEDNRBALDH1A1MAPK1
SCHEMBL7426853 0.77 SLC22A12 (0.40) SLC22A12CA12CA1CA2CA9
SCHEMBL7423537 0.75 MEN1 (0.40) SLC22A12EDNRAALDH1A1MAPK1LMNA
SCHEMBL7473906 0.74 ALDH1A1 (0.43) SLC22A12EDNRAEDNRBALDH1A1MAPK1
SCHEMBL7707720 0.72 FABP4 (0.48) SLC22A12EDNRAEDNRBALDH1A1MAPK1
SCHEMBL7426960 0.72 ALDH1A1 (0.51) SLC22A12EDNRAEDNRBALDH1A1MAPK1
SCHEMBL7425503 0.70 EDNRA (0.41) SLC22A12EDNRAEDNRBALDH1A1MAPK1
SCHEMBL7418953 0.70 EDNRA (0.39) SLC22A12EDNRAEDNRBALDH1A1
SCHEMBL7419529 0.70 TP53 (0.49) SLC22A12MAPK8ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6358992-B1 Method of inhibiting neoplastic cells with indole derivatives CELL PATHWAYS, INC. 2002-03-19 US disclosed