SCHEMBL7722089

SCHEMBL7722089

Cc1c(Cl)cccc1N1CCN(C(=O)[C@H]2C[C@H](NC(=O)[C@@H](O)CNC(=O)OC(C)(C)C)CN2C(=O)OC(C)(C)C)CC1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 1/20 0.42
LMNA P02545 4/20 0.40
DRD2 P14416 5/20 0.39
DRD3 P35462 1/20 0.39
TP53 P04637 2/20 0.37
HTR2A P28223 3/20 0.37
HTR2C P28335 3/20 0.37
SLC6A4 P31645 3/20 0.37
ADAM17 P78536 1/20 0.35
ADAMTS5 Q9UNA0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7722092 0.84 LMNA (0.40) TGM2LMNADRD2DRD3TP53
SCHEMBL7728458 0.83 DRD2 (0.51) TGM2LMNADRD2DRD3TP53
SCHEMBL7728454 0.83 DRD2 (0.51) TGM2LMNADRD2DRD3TP53
SCHEMBL7722007 0.81 TGM2 (0.42) TGM2LMNADRD2DRD3TP53
SCHEMBL7722003 0.81 TGM2 (0.42) TGM2LMNADRD2DRD3TP53
SCHEMBL7722009 0.81 TGM2 (0.42) TGM2LMNADRD2DRD3TP53
SCHEMBL7729067 0.76 BTK (0.38)
SCHEMBL7728349 0.76 BTK (0.38)
SCHEMBL7727553 0.76 BTK (0.38)
SCHEMBL7728341 0.76 BTK (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399629-B1 PYRROLIDINES AND PIPERIDINES FOR TREATING MICROBIAL INFECTIONS BY REDUCING EXPORT OF COADMINISTERED ANTIMICROBIAL AGENT OR COMPOUND SYNTHESIZED BY MICROBES FOR THEIR GROWTH; REDUCING IN VIVO AVAILABILITY MICROCIDE PHARMACEUTICALS, INC. 2002-06-04 US disclosed
WO-2000001714-A1 EFFLUX PUMP INHIBITORS MICROCIDE PHARMACEUTICALS, INC. (US) 2000-01-13 WO disclosed